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1,5-Disubstituted Acylated 2-Amino-4,5-dihydroimidazoles as a New Class of Retinoic Acid Receptor-Related Orphan Receptor (ROR) Inhibitors.
Int J Mol Sci. 2022 Apr 17;23(8):4433. doi: 10.3390/ijms23084433.
Int J Mol Sci. 2022.
PMID: 35457251
Free PMC article.
Antinociceptive activity of thiazole-containing cyclized DAMGO and Leu-(Met) enkephalin analogs.
Harris HM, Eans SO, Ganno ML, Davis JC, Dooley CT, McLaughlin JP, Nefzi A.
Harris HM, et al.
Org Biomol Chem. 2019 Jun 7;17(21):5305-5315. doi: 10.1039/c9ob00882a. Epub 2019 May 16.
Org Biomol Chem. 2019.
PMID: 31094391
Free PMC article.
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Synthesis of dihydroimidazole tethered imidazolinethiones and their activity as novel antagonists of the nuclear retinoic acid receptor-related orphan receptors (RORs).
Nefzi A, Marconi GD, Ortiz MA, Davis JC, Piedrafita FJ.
Nefzi A, et al.
Bioorg Med Chem Lett. 2017 Apr 1;27(7):1608-1610. doi: 10.1016/j.bmcl.2017.02.014. Epub 2017 Feb 10.
Bioorg Med Chem Lett. 2017.
PMID: 28242276
Free PMC article.
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Diversity oriented synthesis and IKK inhibition of aminobenzimidazole tethered quinazoline-2,4-diones, thioxoquinazolin-4-ones, benzodiazepine-2,3,5-triones, isoxazoles and isoxazolines.
Dadiboyena S, Arfaoui A, Amri H, Piedrafita FJ, Nefzi A.
Dadiboyena S, et al.
Bioorg Med Chem Lett. 2015 Feb 1;25(3):685-9. doi: 10.1016/j.bmcl.2014.11.078. Epub 2014 Dec 8.
Bioorg Med Chem Lett. 2015.
PMID: 25522820
Free PMC article.
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