Provins L - Search Results

1

Discovery and development of SV2A PET tracers: Potential for imaging synaptic density and clinical applications.

Mercier J, Provins L, Valade A. Mercier J, et al. Among authors: provins l. Drug Discov Today Technol. 2017 Nov;25:45-52. doi: 10.1016/j.ddtec.2017.11.003. Epub 2017 Dec 1. Drug Discov Today Technol. 2017. PMID: 29233267 Review.

2

Discovery of heterocyclic nonacetamide synaptic vesicle protein 2A (SV2A) ligands with single-digit nanomolar potency: opening avenues towards the first SV2A positron emission tomography (PET) ligands.

Mercier J, Archen L, Bollu V, Carré S, Evrard Y, Jnoff E, Kenda B, Lallemand B, Michel P, Montel F, Moureau F, Price N, Quesnel Y, Sauvage X, Valade A, Provins L. Mercier J, et al. Among authors: provins l. ChemMedChem. 2014 Apr;9(4):693-8. doi: 10.1002/cmdc.201300482. Epub 2014 Jan 20. ChemMedChem. 2014. PMID: 24446373

3

[(11)C]UCB-A, a novel PET tracer for synaptic vesicle protein 2A.

Estrada S, Lubberink M, Thibblin A, Sprycha M, Buchanan T, Mestdagh N, Kenda B, Mercier J, Provins L, Gillard M, Tytgat D, Antoni G. Estrada S, et al. Among authors: provins l. Nucl Med Biol. 2016 Jun;43(6):325-32. doi: 10.1016/j.nucmedbio.2016.03.004. Epub 2016 Mar 17. Nucl Med Biol. 2016. PMID: 27260773

4

Novel Strategies To Activate the Dopamine D₁ Receptor: Recent Advances in Orthosteric Agonism and Positive Allosteric Modulation.

Hall A, Provins L, Valade A. Hall A, et al. Among authors: provins l. J Med Chem. 2019 Jan 10;62(1):128-140. doi: 10.1021/acs.jmedchem.8b01767. Epub 2018 Dec 27. J Med Chem. 2019. PMID: 30525590 Review.

5

Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists.

Provins L, Denonne F, Célanire S, Christophe B, Defays S, Delaunoy C, Delporte ML, Demaude T, Durieu V, Gillard M, Hubert D, Lamberty Y, Lorent G, Valade A, Vanbellinghen A, Van Houtvin N. Provins L, et al. ChemMedChem. 2012 Dec;7(12):2087-92. doi: 10.1002/cmdc.201200406. Epub 2012 Oct 5. ChemMedChem. 2012. PMID: 23042668

6

Back-up strategies in drug discovery: what, how and when?

Provins L, Jnoff E, Genicot C. Provins L, et al. Drug Discov Today. 2014 Nov;19(11):1808-1811. doi: 10.1016/j.drudis.2014.07.001. Epub 2014 Jul 10. Drug Discov Today. 2014. PMID: 25017046 Review.

7

Pharmacological Profile of the Novel Antiepileptic Drug Candidate Padsevonil: Interactions with Synaptic Vesicle 2 Proteins and the GABA_A Receptor.

Wood M, Daniels V, Provins L, Wolff C, Kaminski RM, Gillard M. Wood M, et al. Among authors: provins l. J Pharmacol Exp Ther. 2020 Jan;372(1):1-10. doi: 10.1124/jpet.119.261149. Epub 2019 Oct 16. J Pharmacol Exp Ther. 2020. PMID: 31619465

8

Functional characterization of the antiepileptic drug candidate, padsevonil, on GABA_A receptors.

Niespodziany I, Ghisdal P, Mullier B, Wood M, Provins L, Kaminski RM, Wolff C. Niespodziany I, et al. Among authors: provins l. Epilepsia. 2020 May;61(5):914-923. doi: 10.1111/epi.16497. Epub 2020 Apr 16. Epilepsia. 2020. PMID: 32297665 Free PMC article.

9

Pharmacological Profile of the Novel Antiepileptic Drug Candidate Padsevonil: Characterization in Rodent Seizure and Epilepsy Models.

Leclercq K, Matagne A, Provins L, Klitgaard H, Kaminski RM. Leclercq K, et al. Among authors: provins l. J Pharmacol Exp Ther. 2020 Jan;372(1):11-20. doi: 10.1124/jpet.119.261222. Epub 2019 Oct 16. J Pharmacol Exp Ther. 2020. PMID: 31619464

10

Discovery of a new class of non-imidazole oxazoline-based histamine H(3) receptor (H(3)R) inverse agonists.

Célanire S, Wijtmans M, Christophe B, Collart P, de Esch I, Dassesse D, Delaunoy C, Denonne F, Durieu V, Gelens E, Gillard M, Lallemand B, Lamberty Y, Lebon F, Nicolas JM, Quéré L, Snip E, Vanbellinghen A, Van Houtvin N, Verbois V, Timmerman H, Talaga P, Leurs R, Provins L. Célanire S, et al. Among authors: provins l. ChemMedChem. 2009 Jul;4(7):1063-8. doi: 10.1002/cmdc.200900055. ChemMedChem. 2009. PMID: 19405064

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