Previti S - Search Results

1

Design and evaluation of non-carboxylate 5-arylidene-2-thioxo-4-imidazolidinones as novel non-competitive inhibitors of protein tyrosine phosphatase 1B.

Ottanà R, Paoli P, Lori G, Adornato I, Previti S, Naß A, Wolber G, Maccari R. Ottanà R, et al. Among authors: previti s. Bioorg Chem. 2019 Nov;92:103211. doi: 10.1016/j.bioorg.2019.103211. Epub 2019 Aug 21. Bioorg Chem. 2019. PMID: 31491569

2

Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation.

Ettari R, Pinto A, Previti S, Tamborini L, Angelo IC, La Pietra V, Marinelli L, Novellino E, Schirmeister T, Zappalà M, Grasso S, De Micheli C, Conti P. Ettari R, et al. Among authors: previti s. Bioorg Med Chem. 2015 Nov 1;23(21):7053-60. doi: 10.1016/j.bmc.2015.09.029. Epub 2015 Sep 21. Bioorg Med Chem. 2015. PMID: 26432608

3

Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agents.

Ettari R, Previti S, Cosconati S, Maiorana S, Schirmeister T, Grasso S, Zappalà M. Ettari R, et al. Among authors: previti s. Bioorg Med Chem Lett. 2016 Aug 1;26(15):3453-6. doi: 10.1016/j.bmcl.2016.06.047. Epub 2016 Jun 21. Bioorg Med Chem Lett. 2016. PMID: 27372809

4

Identification of 2-thioxoimidazolidin-4-one derivatives as novel noncovalent proteasome and immunoproteasome inhibitors.

Maccari R, Ettari R, Adornato I, Naß A, Wolber G, Bitto A, Mannino F, Aliquò F, Bruno G, Nicolò F, Previti S, Grasso S, Zappalà M, Ottanà R. Maccari R, et al. Among authors: previti s. Bioorg Med Chem Lett. 2018 Feb 1;28(3):278-283. doi: 10.1016/j.bmcl.2017.12.053. Epub 2017 Dec 26. Bioorg Med Chem Lett. 2018. PMID: 29292224

5

Development of Novel Benzodiazepine-Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense.

Di Chio C, Previti S, Amendola G, Cosconati S, Schirmeister T, Zappalà M, Ettari R. Di Chio C, et al. Among authors: previti s. ChemMedChem. 2020 Jun 4;15(11):995-1001. doi: 10.1002/cmdc.202000158. Epub 2020 May 5. ChemMedChem. 2020. PMID: 32329206

6

Development of isoquinolinone derivatives as immunoproteasome inhibitors.

Ettari R, Iraci N, Di Chio C, Previti S, Danzè M, Zappalà M. Ettari R, et al. Among authors: previti s. Bioorg Med Chem Lett. 2022 Jan 1;55:128478. doi: 10.1016/j.bmcl.2021.128478. Epub 2021 Nov 24. Bioorg Med Chem Lett. 2022. PMID: 34838650

7

Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense.

Di Chio C, Previti S, Amendola G, Ravichandran R, Wagner A, Cosconati S, Hellmich UA, Schirmeister T, Zappalà M, Ettari R. Di Chio C, et al. Among authors: previti s. Eur J Med Chem. 2022 Jun 5;236:114328. doi: 10.1016/j.ejmech.2022.114328. Epub 2022 Mar 29. Eur J Med Chem. 2022. PMID: 35385806

8

Influence of amino acid size at the P3 position of N-Cbz-tripeptide Michael acceptors targeting falcipain-2 and rhodesain for the treatment of malaria and human african trypanosomiasis.

Previti S, Ettari R, Di Chio C, Legac J, Bogacz M, Zimmer C, Schirmeister T, Rosenthal PJ, Zappalà M. Previti S, et al. Bioorg Chem. 2023 Aug;137:106587. doi: 10.1016/j.bioorg.2023.106587. Epub 2023 May 4. Bioorg Chem. 2023. PMID: 37163812 Free article.

9

Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs).

Previti S, Ettari R, Cosconati S, Amendola G, Chouchene K, Wagner A, Hellmich UA, Ulrich K, Krauth-Siegel RL, Wich PR, Schmid I, Schirmeister T, Gut J, Rosenthal PJ, Grasso S, Zappalà M. Previti S, et al. J Med Chem. 2017 Aug 24;60(16):6911-6923. doi: 10.1021/acs.jmedchem.7b00405. Epub 2017 Aug 11. J Med Chem. 2017. PMID: 28763614

10

Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis.

Ettari R, Previti S, Maiorana S, Amendola G, Wagner A, Cosconati S, Schirmeister T, Hellmich UA, Zappalà M. Ettari R, et al. Among authors: previti s. J Med Chem. 2019 Dec 12;62(23):10617-10629. doi: 10.1021/acs.jmedchem.9b00908. Epub 2019 Nov 27. J Med Chem. 2019. PMID: 31714776

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