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Identification of potent tricyclic prodrug S1P1 receptor modulators.
Medchemcomm. 2016 Nov 25;8(4):725-729. doi: 10.1039/c6md00539j. eCollection 2017 Apr 1.
Medchemcomm. 2016.
PMID: 30108791
Free PMC article.
Identification and Preclinical Pharmacology of ((1 R,3 S)-1-Amino-3-(( S)-6-(2-methoxyphenethyl)-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986166): A Differentiated Sphingosine-1-phosphate Receptor 1 (S1P1) Modulator Advanced into Clinical Trials.
Gilmore JL, Xiao HY, Dhar TGM, Yang MG, Xiao Z, Xie J, Lehman-McKeeman LD, Gong L, Sun H, Lecureux L, Chen C, Wu DR, Dabros M, Yang X, Taylor TL, Zhou XD, Heimrich EM, Thomas R, McIntyre KW, Borowski V, Warrack BM, Li Y, Shi H, Levesque PC, Yang Z, Marino AM, Cornelius G, D'Arienzo CJ, Mathur A, Rampulla R, Gupta A, Pragalathan B, Shen DR, Cvijic ME, Salter-Cid LM, Carter PH, Dyckman AJ.
Gilmore JL, et al. Among authors: pragalathan b.
J Med Chem. 2019 Mar 14;62(5):2265-2285. doi: 10.1021/acs.jmedchem.8b01695. Epub 2019 Mar 6.
J Med Chem. 2019.
PMID: 30785748
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Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P1 Receptor Modulator.
Yang MG, Xiao Z, Dhar TG, Xiao HY, Gilmore JL, Marcoux D, Xie JH, McIntyre KW, Taylor TL, Borowski V, Heimrich E, Li YW, Feng J, Fernandes A, Yang Z, Balimane P, Marino AM, Cornelius G, Warrack BM, Mathur A, Wu DR, Li P, Gupta A, Pragalathan B, Shen DR, Cvijic ME, Lehman-McKeeman LD, Salter-Cid L, Barrish JC, Carter PH, Dyckman AJ.
Yang MG, et al. Among authors: pragalathan b.
J Med Chem. 2016 Dec 22;59(24):11138-11147. doi: 10.1021/acs.jmedchem.6b01433. Epub 2016 Dec 7.
J Med Chem. 2016.
PMID: 28002964
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Discovery of a Highly Selective JAK2 Inhibitor, BMS-911543, for the Treatment of Myeloproliferative Neoplasms.
Wan H, Schroeder GM, Hart AC, Inghrim J, Grebinski J, Tokarski JS, Lorenzi MV, You D, Mcdevitt T, Penhallow B, Vuppugalla R, Zhang Y, Gu X, Iyer R, Lombardo LJ, Trainor GL, Ruepp S, Lippy J, Blat Y, Sack JS, Khan JA, Stefanski K, Sleczka B, Mathur A, Sun JH, Wong MK, Wu DR, Li P, Gupta A, Arunachalam PN, Pragalathan B, Narayanan S, K C N, Kuppusamy P, Purandare AV.
Wan H, et al. Among authors: pragalathan b.
ACS Med Chem Lett. 2015 Jul 12;6(8):850-5. doi: 10.1021/acsmedchemlett.5b00226. eCollection 2015 Aug 13.
ACS Med Chem Lett. 2015.
PMID: 26288683
Free PMC article.
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Pancreatic Non-Hodgkin Lymphoma, a rare cause for obstructive jaundice. A Case reports.
B P, K I, A A J, S G.
B P, et al.
Int J Surg Case Rep. 2021 Jan;78:369-371. doi: 10.1016/j.ijscr.2020.12.071. Epub 2020 Dec 26.
Int J Surg Case Rep. 2021.
PMID: 33401192
Free PMC article.
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Torsion of an Epididymal Cyst: A Rare Finding on Scrotal Exploration for Acute Scrotum.
Ozaal AMOM, Pragalathan B, Lavanya S, Sarma ST.
Ozaal AMOM, et al. Among authors: pragalathan b.
Case Rep Urol. 2020 Nov 22;2020:8858606. doi: 10.1155/2020/8858606. eCollection 2020.
Case Rep Urol. 2020.
PMID: 33299634
Free PMC article.
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Omental tuberculosis (TB) is a rare disease which can mimic Gastrointestinal malignancies: A case report.
Pragalathan B, Omar Mohamed Ozaal AM, Lavanya S, Raviraj S.
Pragalathan B, et al.
Int J Surg Case Rep. 2020;77:318-320. doi: 10.1016/j.ijscr.2020.10.118. Epub 2020 Oct 30.
Int J Surg Case Rep. 2020.
PMID: 33197776
Free PMC article.
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