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Page 1
Antifungal Thiazolidines: Synthesis and Biological Evaluation of Mycosidine Congeners.
Levshin IB, Simonov AY, Lavrenov SN, Panov AA, Grammatikova NE, Alexandrov AA, Ghazy ESMO, Savin NA, Gorelkin PV, Erofeev AS, Polshakov VI. Levshin IB, et al. Among authors: polshakov vi. Pharmaceuticals (Basel). 2022 May 1;15(5):563. doi: 10.3390/ph15050563. Pharmaceuticals (Basel). 2022. PMID: 35631390 Free PMC article.
Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them.
Machulkin AE, Shafikov RR, Uspenskaya AA, Petrov SA, Ber AP, Skvortsov DA, Nimenko EA, Zyk NU, Smirnova GB, Pokrovsky VS, Abakumov MA, Saltykova IV, Akhmirov RT, Garanina AS, Polshakov VI, Saveliev OY, Ivanenkov YA, Aladinskaya AV, Finko AV, Yamansarov EU, Krasnovskaya OO, Erofeev AS, Gorelkin PV, Dontsova OA, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: polshakov vi. J Med Chem. 2021 Apr 22;64(8):4532-4552. doi: 10.1021/acs.jmedchem.0c01935. Epub 2021 Apr 6. J Med Chem. 2021. PMID: 33822606
Synthesis, Characterization, and Preclinical Evaluation of a Small-Molecule Prostate-Specific Membrane Antigen-Targeted Monomethyl Auristatin E Conjugate.
Machulkin AE, Uspenskaya AA, Zyk NU, Nimenko EA, Ber AP, Petrov SA, Polshakov VI, Shafikov RR, Skvortsov DA, Plotnikova EA, Pankratov AA, Smirnova GB, Borisova YA, Pokrovsky VS, Kolmogorov VS, Vaneev AN, Khudyakov AD, Chepikova OE, Kovalev S, Zamyatnin AA Jr, Erofeev A, Gorelkin P, Beloglazkina EK, Zyk NV, Khazanova ES, Majouga AG. Machulkin AE, et al. Among authors: polshakov vi. J Med Chem. 2021 Dec 9;64(23):17123-17145. doi: 10.1021/acs.jmedchem.1c01157. Epub 2021 Nov 19. J Med Chem. 2021. PMID: 34797052
Polypeptide-Based Molecular Platform and Its Docetaxel/Sulfo-Cy5-Containing Conjugate for Targeted Delivery to Prostate Specific Membrane Antigen.
Petrov SA, Machulkin AE, Uspenskaya AA, Zyk NY, Nimenko EA, Garanina AS, Petrov RA, Polshakov VI, Grishin YK, Roznyatovsky VA, Zyk NV, Majouga AG, Beloglazkina EK. Petrov SA, et al. Among authors: polshakov vi. Molecules. 2020 Dec 8;25(24):5784. doi: 10.3390/molecules25245784. Molecules. 2020. PMID: 33302417 Free PMC article.
Conjugates of Chloramphenicol Amine and Berberine as Antimicrobial Agents.
Pavlova JA, Tereshchenkov AG, Nazarov PA, Lukianov DA, Skvortsov DA, Polshakov VI, Vasilieva BF, Efremenkova OV, Kaiumov MY, Paleskava A, Konevega AL, Dontsova OA, Osterman IA, Bogdanov AA, Sumbatyan NV. Pavlova JA, et al. Among authors: polshakov vi. Antibiotics (Basel). 2022 Dec 22;12(1):15. doi: 10.3390/antibiotics12010015. Antibiotics (Basel). 2022. PMID: 36671216 Free PMC article.
Biological evaluation and spectral characterization of a novel tetracenomycin X congener.
Alferova VA, Maviza TP, Biryukov MV, Zakalyukina YV, Lukianov DA, Skvortsov DA, Vasilyeva LA, Tashlitsky VN, Polshakov VI, Sergiev PV, Korshun VA, Osterman IA. Alferova VA, et al. Among authors: polshakov vi. Biochimie. 2022 Jan;192:63-71. doi: 10.1016/j.biochi.2021.09.014. Epub 2021 Sep 28. Biochimie. 2022. PMID: 34592388
NMR assignments of the WBSCR27 protein related to Williams-Beuren syndrome.
Mariasina SS, Petrova OA, Osterman IA, Sergeeva OV, Efimov SV, Klochkov VV, Sergiev PV, Dontsova OA, Huang TH, Chang CF, Polshakov VI. Mariasina SS, et al. Among authors: polshakov vi. Biomol NMR Assign. 2018 Oct;12(2):303-308. doi: 10.1007/s12104-018-9827-2. Epub 2018 Jun 4. Biomol NMR Assign. 2018. PMID: 29868988
69 results