Pinna GA - Search Results

1

Synthesis and SAR study of novel tricyclic pyrazoles as potent phosphodiesterase 10A inhibitors.

Dore A, Asproni B, Scampuddu A, Pinna GA, Christoffersen CT, Langgård M, Kehler J. Dore A, et al. Among authors: pinna ga. Eur J Med Chem. 2014 Sep 12;84:181-93. doi: 10.1016/j.ejmech.2014.07.020. Epub 2014 Jul 7. Eur J Med Chem. 2014. PMID: 25016376

2

N-3(9)-arylpropenyl-N-9(3)-propionyl-3,9-diazabicyclo[3.3.1]nonanes as mu-opioid receptor agonists. Effects on mu-affinity of arylalkenyl chain modifications.

Pinna GA, Cignarella G, Loriga G, Murineddu G, Mussinu JM, Ruiu S, Fadda P, Fratta W. Pinna GA, et al. Bioorg Med Chem. 2002 Jun;10(6):1929-37. doi: 10.1016/s0968-0896(01)00436-9. Bioorg Med Chem. 2002. PMID: 11937351

3

Tricyclic pyrazoles. Part 1: synthesis and biological evaluation of novel 1,4-dihydroindeno[1,2-c]pyrazol-based ligands for CB1and CB2 cannabinoid receptors.

Mussinu JM, Ruiu S, Mulè AC, Pau A, Carai MA, Loriga G, Murineddu G, Pinna GA. Mussinu JM, et al. Among authors: pinna ga. Bioorg Med Chem. 2003 Jan 17;11(2):251-63. doi: 10.1016/s0968-0896(02)00319-x. Bioorg Med Chem. 2003. PMID: 12470719

4

Synthesis of novel diazatricyclodecanes (DTDs). Effects of structural variation at the C3' allyl end and at the phenyl ring of the cinnamyl chain on mu-receptor affinity and opioid antinociception.

Pinna GA, Cignarella G, Ruiu S, Loriga G, Murineddu G, Villa S, Grella GE, Cossu G, Fratta W. Pinna GA, et al. Bioorg Med Chem. 2003 Sep 1;11(18):4015-26. doi: 10.1016/s0968-0896(03)00373-0. Bioorg Med Chem. 2003. PMID: 12927864

5

Tricyclic pyrazoles. Part 2: Synthesis and biological evaluation of novel 4,5-dihydro-1H-benzo[g]indazole-based ligands for cannabinoid receptors.

Murineddu G, Ruiu S, Mussinu JM, Loriga G, Grella GE, Carai MA, Lazzari P, Pani L, Pinna GA. Murineddu G, et al. Among authors: pinna ga. Bioorg Med Chem. 2005 May 2;13(9):3309-20. doi: 10.1016/j.bmc.2005.02.032. Bioorg Med Chem. 2005. PMID: 15809166

6

Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for the opioid receptors.

Loriga G, Manca I, Murineddu G, Chelucci G, Villa S, Gessi S, Toma L, Cignarella G, Pinna GA. Loriga G, et al. Among authors: pinna ga. Bioorg Med Chem. 2006 Feb 1;14(3):676-91. doi: 10.1016/j.bmc.2005.09.045. Epub 2005 Oct 20. Bioorg Med Chem. 2006. PMID: 16243530

7

Tricyclic pyrazoles. 3. Synthesis, biological evaluation, and molecular modeling of analogues of the cannabinoid antagonist 8-chloro-1-(2',4'-dichlorophenyl)-N-piperidin-1-yl-1,4,5,6-tetrahydrobenzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide.

Murineddu G, Ruiu S, Loriga G, Manca I, Lazzari P, Reali R, Pani L, Toma L, Pinna GA. Murineddu G, et al. Among authors: pinna ga. J Med Chem. 2005 Nov 17;48(23):7351-62. doi: 10.1021/jm050317f. J Med Chem. 2005. PMID: 16279795

8

Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide.

Murineddu G, Lazzari P, Ruiu S, Sanna A, Loriga G, Manca I, Falzoi M, Dessì C, Curzu MM, Chelucci G, Pani L, Pinna GA. Murineddu G, et al. Among authors: pinna ga. J Med Chem. 2006 Dec 14;49(25):7502-12. doi: 10.1021/jm060920d. J Med Chem. 2006. PMID: 17149879

9

3-{2-[Bis-(4-fluorophenyl)methoxy]ethyl}-6-substituted-3,6-diazabicyclo[3.1.1]heptanes as novel potent dopamine uptake inhibitors.

Loriga G, Ruiu S, Manca I, Murineddu G, Dessi C, Pani L, Pinna GA. Loriga G, et al. Among authors: pinna ga. Bioorg Med Chem. 2007 Jun 1;15(11):3748-55. doi: 10.1016/j.bmc.2007.03.035. Epub 2007 Mar 16. Bioorg Med Chem. 2007. PMID: 17399987

10

Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptors.

Murineddu G, Murruzzu C, Curzu MM, Chelucci G, Gotti C, Gaimarri A, Legnani L, Toma L, Pinna GA. Murineddu G, et al. Among authors: pinna ga. Bioorg Med Chem Lett. 2008 Dec 1;18(23):6147-50. doi: 10.1016/j.bmcl.2008.10.002. Epub 2008 Oct 5. Bioorg Med Chem Lett. 2008. PMID: 18938077

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