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Anti-Plasmodium falciparum activity of quinoline-sulfonamide hybrids.
Pinheiro LC, Boechat N, Ferreira Mde L, Júnior CC, Jesus AM, Leite MM, Souza NB, Krettli AU. Pinheiro LC, et al. Bioorg Med Chem. 2015 Sep 1;23(17):5979-84. doi: 10.1016/j.bmc.2015.06.056. Epub 2015 Jul 2. Bioorg Med Chem. 2015. PMID: 26190461
SAR of a series of anti-HSV-1 acridone derivatives, and a rational acridone-based design of a new anti-HSV-1 3H-benzo[b]pyrazolo[3,4-h]-1,6-naphthyridine series.
Bernardino AM, Castro HC, Frugulhetti IC, Loureiro NI, Azevedo AR, Pinheiro LC, Souza TM, Giongo V, Passamani F, Magalhães UO, Albuquerque MG, Cabral LM, Rodrigues CR. Bernardino AM, et al. Among authors: pinheiro lc. Bioorg Med Chem. 2008 Jan 1;16(1):313-21. doi: 10.1016/j.bmc.2007.09.032. Epub 2007 Sep 22. Bioorg Med Chem. 2008. PMID: 17937990
New trifluoromethyl triazolopyrimidines as anti-Plasmodium falciparum agents.
Boechat N, Pinheiro LC, Silva TS, Aguiar AC, Carvalho AS, Bastos MM, Costa CC, Pinheiro S, Pinto AC, Mendonça JS, Dutra KD, Valverde AL, Santos-Filho OA, Ceravolo IP, Krettli AU. Boechat N, et al. Among authors: pinheiro s, pinheiro lc. Molecules. 2012 Jul 10;17(7):8285-302. doi: 10.3390/molecules17078285. Molecules. 2012. PMID: 22781441 Free PMC article.
Novel selective inhibitor of Leishmania (Leishmania) amazonensis arginase.
da Silva ER, Boechat N, Pinheiro LC, Bastos MM, Costa CC, Bartholomeu JC, da Costa TH. da Silva ER, et al. Among authors: pinheiro lc. Chem Biol Drug Des. 2015 Nov;86(5):969-78. doi: 10.1111/cbdd.12566. Epub 2015 May 14. Chem Biol Drug Des. 2015. PMID: 25845502
249 results