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Enzymatic Preparation of 2'-5',3'-5'-Cyclic Dinucleotides, Their Binding Properties to Stimulator of Interferon Genes Adaptor Protein, and Structure/Activity Correlations.
J Med Chem. 2019 Dec 12;62(23):10676-10690. doi: 10.1021/acs.jmedchem.9b01062. Epub 2019 Nov 27.
J Med Chem. 2019.
PMID: 31715099
Synthesis and Biological Evaluation of Phosphoester and Phosphorothioate Prodrugs of STING Agonist 3',3'-c-Di(2'F,2'dAMP).
Pimková Polidarová M, Břehová P, Kaiser MM, Smola M, Dračínský M, Smith J, Marek A, Dejmek M, Šála M, Gutten O, Rulíšek L, Novotná B, Brázdová A, Janeba Z, Nencka R, Boura E, Páv O, Birkuš G.
Pimková Polidarová M, et al.
J Med Chem. 2021 Jun 10;64(11):7596-7616. doi: 10.1021/acs.jmedchem.1c00301. Epub 2021 May 21.
J Med Chem. 2021.
PMID: 34019405
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STING Agonist-Mediated Cytokine Secretion Is Accompanied by Monocyte Apoptosis.
Pimkova Polidarova M, Brehova P, Dejmek M, Birkus G, Brazdova A.
Pimkova Polidarova M, et al.
ACS Infect Dis. 2022 Mar 11;8(3):463-471. doi: 10.1021/acsinfecdis.1c00554. Epub 2022 Feb 8.
ACS Infect Dis. 2022.
PMID: 35132859
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Synthetic Stimulator of Interferon Genes (STING) Agonists Induce a Cytokine-Mediated Anti-Hepatitis B Virus Response in Nonparenchymal Liver Cells.
Pimkova Polidarova M, Vanekova L, Brehova P, Dejmek M, Vavrina Z, Birkus G, Brazdova A.
Pimkova Polidarova M, et al.
ACS Infect Dis. 2023 Jan 13;9(1):23-32. doi: 10.1021/acsinfecdis.2c00424. Epub 2022 Dec 6.
ACS Infect Dis. 2023.
PMID: 36472628
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