Piersanti G - Search Results

1

Synthesis of benzo[1,2-d;3,4-d']diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists.

Piersanti G, Giorgi L, Bartoccini F, Tarzia G, Minetti P, Gallo G, Giorgi F, Castorina M, Ghirardi O, Carminati P. Piersanti G, et al. Org Biomol Chem. 2007 Aug 21;5(16):2567-71. doi: 10.1039/b707599e. Org Biomol Chem. 2007. PMID: 18019530

2

Design, synthesis, and structure-activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors.

Tarzia G, Duranti A, Tontini A, Piersanti G, Mor M, Rivara S, Plazzi PV, Park C, Kathuria S, Piomelli D. Tarzia G, et al. Among authors: piersanti g. J Med Chem. 2003 Jun 5;46(12):2352-60. doi: 10.1021/jm021119g. J Med Chem. 2003. PMID: 12773040 Free article.

3

5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT) and related compounds induce apoptotic patterns in cultures of human tumor cell lines.

Burattini S, Luchetti F, Battistelli M, Della Felice M, Papa S, Piersanti G, Tarzia G, Falcieri E. Burattini S, et al. Among authors: piersanti g. J Biol Regul Homeost Agents. 2003 Oct-Dec;17(4):348-57. J Biol Regul Homeost Agents. 2003. PMID: 15065766

4

Strategies leading to MT2 selective melatonin receptor antagonists.

Spadoni G, Bedini A, Piersanti G, Mor M, Rivara S, Tarzia G. Spadoni G, et al. Among authors: piersanti g. Adv Exp Med Biol. 2003;527:577-85. doi: 10.1007/978-1-4615-0135-0_66. Adv Exp Med Biol. 2003. PMID: 15206776

5

Tricyclic alkylamides as melatonin receptor ligands with antagonist or inverse agonist activity.

Lucini V, Pannacci M, Scaglione F, Fraschini F, Rivara S, Mor M, Bordi F, Plazzi PV, Spadoni G, Bedini A, Piersanti G, Diamantini G, Tarzia G. Lucini V, et al. Among authors: piersanti g. J Med Chem. 2004 Aug 12;47(17):4202-12. doi: 10.1021/jm040768k. J Med Chem. 2004. PMID: 15293992

6

Cyclohexylcarbamic acid 3'- or 4'-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: synthesis, quantitative structure-activity relationships, and molecular modeling studies.

Mor M, Rivara S, Lodola A, Plazzi PV, Tarzia G, Duranti A, Tontini A, Piersanti G, Kathuria S, Piomelli D. Mor M, et al. Among authors: piersanti g. J Med Chem. 2004 Oct 7;47(21):4998-5008. doi: 10.1021/jm031140x. J Med Chem. 2004. PMID: 15456244 Free article.

7

2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.

Minetti P, Tinti MO, Carminati P, Castorina M, Di Cesare MA, Di Serio S, Gallo G, Ghirardi O, Giorgi F, Giorgi L, Piersanti G, Bartoccini F, Tarzia G. Minetti P, et al. Among authors: piersanti g. J Med Chem. 2005 Nov 3;48(22):6887-96. doi: 10.1021/jm058018d. J Med Chem. 2005. PMID: 16250647

8

Synthesis and structure-activity relationships of FAAH inhibitors: cyclohexylcarbamic acid biphenyl esters with chemical modulation at the proximal phenyl ring.

Tarzia G, Duranti A, Gatti G, Piersanti G, Tontini A, Rivara S, Lodola A, Plazzi PV, Mor M, Kathuria S, Piomelli D. Tarzia G, et al. Among authors: piersanti g. ChemMedChem. 2006 Jan;1(1):130-9. doi: 10.1002/cmdc.200500017. ChemMedChem. 2006. PMID: 16892344

9

An improved synthesis of cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT(2) melatonin receptor antagonist.

Lucarini S, Bedini A, Spadoni G, Piersanti G. Lucarini S, et al. Among authors: piersanti g. Org Biomol Chem. 2008 Jan 7;6(1):147-50. doi: 10.1039/b713904g. Epub 2007 Nov 13. Org Biomol Chem. 2008. PMID: 18075659

10

Synthesis and quantitative structure-activity relationship of fatty acid amide hydrolase inhibitors: modulation at the N-portion of biphenyl-3-yl alkylcarbamates.

Mor M, Lodola A, Rivara S, Vacondio F, Duranti A, Tontini A, Sanchini S, Piersanti G, Clapper JR, King AR, Tarzia G, Piomelli D. Mor M, et al. Among authors: piersanti g. J Med Chem. 2008 Jun 26;51(12):3487-98. doi: 10.1021/jm701631z. Epub 2008 May 29. J Med Chem. 2008. PMID: 18507372 Free PMC article.

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