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Alkoxycarbonate Ester Prodrugs of Preclinical Drug Candidate ELQ-300 for Prophylaxis and Treatment of Malaria.
ACS Infect Dis. 2017 Oct 13;3(10):728-735. doi: 10.1021/acsinfecdis.7b00062. Epub 2017 Sep 27.
ACS Infect Dis. 2017.
PMID: 28927276
Free PMC article.
Discovery, synthesis, and optimization of antimalarial 4(1H)-quinolone-3-diarylethers.
Nilsen A, Miley GP, Forquer IP, Mather MW, Katneni K, Li Y, Pou S, Pershing AM, Stickles AM, Ryan E, Kelly JX, Doggett JS, White KL, Hinrichs DJ, Winter RW, Charman SA, Zakharov LN, Bathurst I, Burrows JN, Vaidya AB, Riscoe MK.
Nilsen A, et al. Among authors: pershing am.
J Med Chem. 2014 May 8;57(9):3818-34. doi: 10.1021/jm500147k. Epub 2014 Apr 18.
J Med Chem. 2014.
PMID: 24720377
Free PMC article.
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Inhibition of cytochrome bc1 as a strategy for single-dose, multi-stage antimalarial therapy.
Stickles AM, Ting LM, Morrisey JM, Li Y, Mather MW, Meermeier E, Pershing AM, Forquer IP, Miley GP, Pou S, Winter RW, Hinrichs DJ, Kelly JX, Kim K, Vaidya AB, Riscoe MK, Nilsen A.
Stickles AM, et al. Among authors: pershing am.
Am J Trop Med Hyg. 2015 Jun;92(6):1195-201. doi: 10.4269/ajtmh.14-0553. Epub 2015 Apr 27.
Am J Trop Med Hyg. 2015.
PMID: 25918204
Free PMC article.
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ELQ-300 prodrugs for enhanced delivery and single-dose cure of malaria.
Miley GP, Pou S, Winter R, Nilsen A, Li Y, Kelly JX, Stickles AM, Mather MW, Forquer IP, Pershing AM, White K, Shackleford D, Saunders J, Chen G, Ting LM, Kim K, Zakharov LN, Donini C, Burrows JN, Vaidya AB, Charman SA, Riscoe MK.
Miley GP, et al. Among authors: pershing am.
Antimicrob Agents Chemother. 2015 Sep;59(9):5555-60. doi: 10.1128/AAC.01183-15. Epub 2015 Jun 29.
Antimicrob Agents Chemother. 2015.
PMID: 26124159
Free PMC article.
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ATP synthase complex of Plasmodium falciparum: dimeric assembly in mitochondrial membranes and resistance to genetic disruption.
Nina PB, Morrisey JM, Ganesan SM, Ke H, Pershing AM, Mather MW, Vaidya AB.
Nina PB, et al. Among authors: pershing am.
J Biol Chem. 2011 Dec 2;286(48):41312-41322. doi: 10.1074/jbc.M111.290973. Epub 2011 Oct 7.
J Biol Chem. 2011.
PMID: 21984828
Free PMC article.
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Precision-cut tissue chips as an in vitro toxicology system.
Catania JM, Pershing AM, Gandolfi AJ.
Catania JM, et al. Among authors: pershing am.
Toxicol In Vitro. 2007 Aug;21(5):956-61. doi: 10.1016/j.tiv.2007.02.001. Epub 2007 Feb 13.
Toxicol In Vitro. 2007.
PMID: 17376647
Free PMC article.
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