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Year | Number of Results |
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2016 | 2 |
2018 | 1 |
2019 | 2 |
2020 | 1 |
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2024 | 0 |
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Page 1
Ocular Pharmacokinetics of Intravitreally Injected Protein Therapeutics: Comparison among Standard-of-Care Formats.
Mol Pharm. 2021 Jun 7;18(6):2208-2217. doi: 10.1021/acs.molpharmaceut.0c01218. Epub 2021 May 20.
Mol Pharm. 2021.
PMID: 34014104
Understanding the Half-Life Extension of Intravitreally Administered Antibodies Binding to Ocular Albumin.
Hauri S, Jakubiak P, Fueth M, Dengl S, Belli S, Alvarez-Sánchez R, Caruso A.
Hauri S, et al. Among authors: jakubiak p.
Pharmaceutics. 2020 Aug 26;12(9):810. doi: 10.3390/pharmaceutics12090810.
Pharmaceutics. 2020.
PMID: 32858986
Free PMC article.
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Establishment of an In Vitro-In Vivo Correlation for Melanin Binding and the Extension of the Ocular Half-Life of Small-Molecule Drugs.
Jakubiak P, Cantrill C, Urtti A, Alvarez-Sánchez R.
Jakubiak P, et al.
Mol Pharm. 2019 Dec 2;16(12):4890-4901. doi: 10.1021/acs.molpharmaceut.9b00769. Epub 2019 Nov 12.
Mol Pharm. 2019.
PMID: 31670965
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Influence of Melanin Characteristics on Drug Binding Properties.
Jakubiak P, Lack F, Thun J, Urtti A, Alvarez-Sánchez R.
Jakubiak P, et al.
Mol Pharm. 2019 Jun 3;16(6):2549-2556. doi: 10.1021/acs.molpharmaceut.9b00157. Epub 2019 Apr 30.
Mol Pharm. 2019.
PMID: 30998378
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Understanding Molecular Drivers of Melanin Binding To Support Rational Design of Small Molecule Ophthalmic Drugs.
Jakubiak P, Reutlinger M, Mattei P, Schuler F, Urtti A, Alvarez-Sánchez R.
Jakubiak P, et al.
J Med Chem. 2018 Nov 21;61(22):10106-10115. doi: 10.1021/acs.jmedchem.8b01281. Epub 2018 Nov 13.
J Med Chem. 2018.
PMID: 30398862
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Extension of the dissolution-precipitation model for kinetic elucidation of solvent-mediated polymorphic transformations.
Jakubiak P, Schuler F, Alvarez-Sánchez R.
Jakubiak P, et al.
Eur J Pharm Biopharm. 2016 Dec;109:43-48. doi: 10.1016/j.ejpb.2016.08.019. Epub 2016 Sep 17.
Eur J Pharm Biopharm. 2016.
PMID: 27648958
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Development of a Unified Dissolution and Precipitation Model and Its Use for the Prediction of Oral Drug Absorption.
Jakubiak P, Wagner B, Grimm HP, Petrig-Schaffland J, Schuler F, Alvarez-Sánchez R.
Jakubiak P, et al.
Mol Pharm. 2016 Feb 1;13(2):586-98. doi: 10.1021/acs.molpharmaceut.5b00808. Epub 2016 Jan 5.
Mol Pharm. 2016.
PMID: 26674605
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