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Page 1
Curcumin analogues as possible anti-proliferative & anti-inflammatory agents.
Katsori AM, Chatzopoulou M, Dimas K, Kontogiorgis C, Patsilinakos A, Trangas T, Hadjipavlou-Litina D. Katsori AM, et al. Among authors: patsilinakos a. Eur J Med Chem. 2011 Jul;46(7):2722-35. doi: 10.1016/j.ejmech.2011.03.060. Epub 2011 Apr 5. Eur J Med Chem. 2011. PMID: 21514701
Decreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation.
Chatzopoulou M, Patsilinakos A, Vallianatou T, Prnova MS, Zakelj S, Ragno R, Stefek M, Kristl A, Tsantili-Kakoulidou A, Demopoulos VJ. Chatzopoulou M, et al. Among authors: patsilinakos a. Bioorg Med Chem. 2014 Apr 1;22(7):2194-207. doi: 10.1016/j.bmc.2014.02.016. Epub 2014 Feb 26. Bioorg Med Chem. 2014. PMID: 24630695
Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells.
Zwergel C, Czepukojc B, Evain-Bana E, Xu Z, Stazi G, Mori M, Patsilinakos A, Mai A, Botta B, Ragno R, Bagrel D, Kirsch G, Meiser P, Jacob C, Montenarh M, Valente S. Zwergel C, et al. Among authors: patsilinakos a. Eur J Med Chem. 2017 Jul 7;134:316-333. doi: 10.1016/j.ejmech.2017.04.012. Epub 2017 Apr 10. Eur J Med Chem. 2017. PMID: 28431339
Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3 H)-ones.
Nawrozkij MB, Forgione M, Yablokov AS, Lucidi A, Tomaselli D, Patsilinakos A, Panella C, Hailu GS, Kirillov IA, Badia R, Riveira-Muñoz E, Crespan E, Armijos Rivera JI, Cirilli R, Ragno R, Esté JA, Maga G, Mai A, Rotili D. Nawrozkij MB, et al. Among authors: patsilinakos a. J Med Chem. 2019 Jan 24;62(2):604-621. doi: 10.1021/acs.jmedchem.8b01238. Epub 2018 Dec 20. J Med Chem. 2019. PMID: 30525601
Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors.
Mollica A, Pelliccia S, Famiglini V, Stefanucci A, Macedonio G, Chiavaroli A, Orlando G, Brunetti L, Ferrante C, Pieretti S, Novellino E, Benyhe S, Zador F, Erdei A, Szucs E, Samavati R, Dvrorasko S, Tomboly C, Ragno R, Patsilinakos A, Silvestri R. Mollica A, et al. Among authors: patsilinakos a. J Enzyme Inhib Med Chem. 2017 Dec;32(1):444-451. doi: 10.1080/14756366.2016.1260565. J Enzyme Inhib Med Chem. 2017. PMID: 28097916 Free PMC article.
Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors: The case of trifluoroacetylation.
Papastavrou N, Chatzopoulou M, Ballekova J, Cappiello M, Moschini R, Balestri F, Patsilinakos A, Ragno R, Stefek M, Nicolaou I. Papastavrou N, et al. Among authors: patsilinakos a. Eur J Med Chem. 2017 Apr 21;130:328-335. doi: 10.1016/j.ejmech.2017.02.053. Epub 2017 Feb 24. Eur J Med Chem. 2017. PMID: 28259841
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