Patel N - Search Results

1

SAR and biological evaluation of novel trans-3,4-dimethyl-4-arylpiperidine derivatives as opioid antagonists.

Díaz N, Benvenga M, Emmerson P, Favors R, Mangold M, McKinzie J, Patel N, Peters S, Quimby S, Shannon H, Siegel M, Statnick M, Thomas E, Woodland J, Surface P, Mitch C. Díaz N, et al. Among authors: patel n. Bioorg Med Chem Lett. 2005 Sep 1;15(17):3844-8. doi: 10.1016/j.bmcl.2005.05.123. Bioorg Med Chem Lett. 2005. PMID: 15993591

2

2-Chloro-4-[[(1R,2R)-2-hydroxy-2-methyl-cyclopentyl]amino]-3-methyl-benzonitrile: A Transdermal Selective Androgen Receptor Modulator (SARM) for Muscle Atrophy.

Saeed A, Vaught GM, Gavardinas K, Matthews D, Green JE, Losada PG, Bullock HA, Calvert NA, Patel NJ, Sweetana SA, Krishnan V, Henck JW, Luz JG, Wang Y, Jadhav P. Saeed A, et al. J Med Chem. 2016 Jan 28;59(2):750-5. doi: 10.1021/acs.jmedchem.5b01168. Epub 2016 Jan 7. J Med Chem. 2016. PMID: 26683992

3

Defining Target Engagement Required for Efficacy In Vivo at the Retinoic Acid Receptor-Related Orphan Receptor C2 (RORγt).

Lugar CW, Clarke CA, Morphy R, Rudyk H, Sapmaz S, Stites RE, Vaught GM, Furness K, Broughton HB, Durst GL, Clawson DK, Stout SL, Guo SY, Durbin JD, Stayrook KR, Edmondson DD, Kikly K, New NE, Bina HA, Chambers MG, Shetler P, Chang WY, Chang VC, Barr R, Gough WH, Steele JP, Getman B, Patel N, Mathes BM, Richardson TI. Lugar CW, et al. Among authors: patel n. J Med Chem. 2021 May 13;64(9):5470-5484. doi: 10.1021/acs.jmedchem.0c01918. Epub 2021 Apr 14. J Med Chem. 2021. PMID: 33852312

4

Novel 3-aryl indoles as progesterone receptor antagonists for uterine fibroids.

Richardson TI, Clarke CA, Yu KL, Yee YK, Bleisch TJ, Lopez JE, Jones SA, Hughes NE, Muehl BS, Lugar CW, Moore TL, Shetler PK, Zink RW, Osborne JJ, Montrose-Rafizadeh C, Patel N, Geiser AG, Galvin RJ, Dodge JA. Richardson TI, et al. Among authors: patel n. ACS Med Chem Lett. 2010 Dec 9;2(2):148-53. doi: 10.1021/ml100220b. eCollection 2011 Feb 10. ACS Med Chem Lett. 2010. PMID: 24900294 Free PMC article.

5

Investigation of clinical pharmacokinetic variability of an opioid antagonist through physiologically based absorption modeling.

Ding X, He M, Kulkarni R, Patel N, Zhang X. Ding X, et al. Among authors: patel n. J Pharm Sci. 2013 Aug;102(8):2859-74. doi: 10.1002/jps.23629. Epub 2013 Jun 11. J Pharm Sci. 2013. PMID: 23761048 Clinical Trial.

6

Disposition and metabolism of LY2452473, a selective androgen receptor modulator, in humans.

Yi P, Rehmel JF, Cassidy K, Hadden C, Campanale K, Patel N, Johnson J. Yi P, et al. Among authors: patel n. Drug Metab Dispos. 2012 Dec;40(12):2354-64. doi: 10.1124/dmd.112.047613. Epub 2012 Sep 7. Drug Metab Dispos. 2012. PMID: 22961682

7

Pharmacokinetic comparisons of tail-bleeding with cannula- or retro-orbital bleeding techniques in rats using six marketed drugs.

Hui YH, Huang NH, Ebbert L, Bina H, Chiang A, Maples C, Pritt M, Kern T, Patel N. Hui YH, et al. Among authors: patel n. J Pharmacol Toxicol Methods. 2007 Sep-Oct;56(2):256-64. doi: 10.1016/j.vascn.2007.05.006. Epub 2007 Jun 2. J Pharmacol Toxicol Methods. 2007. PMID: 17618130

8

Evaluation and Optimization of Blood Micro-Sampling Methods: Serial Sampling in a Cross-Over Design from an Individual Mouse.

Patel NJ, Wickremsinhe E, Hui YH, Barr A, Masterson N, Ruterbories K, Weller J, Hanes J, Kern T, Perkins E. Patel NJ, et al. J Pharm Pharm Sci. 2016 Oct-Dec;19(4):496-510. doi: 10.18433/J3NK60. J Pharm Pharm Sci. 2016. PMID: 28057168 Free article.

9

A Semi-Physiologically Based Pharmacokinetic Model Describing the Altered Metabolism of Midazolam Due to Inflammation in Mice.

Varkhede N, Patel N, Chang W, Ruterbories K, Forrest ML. Varkhede N, et al. Among authors: patel n. Pharm Res. 2018 Jun 21;35(8):162. doi: 10.1007/s11095-018-2447-9. Pharm Res. 2018. PMID: 29931580 Free PMC article.

10

Development of a selective androgen receptor modulator for transdermal use in hypogonadal patients.

Krishnan V, Patel NJ, Mackrell JG, Sweetana SA, Bullock H, Ma YL, Waterhouse TH, Yaden BC, Henck J, Zeng QQ, Gavardinas K, Jadhav P, Saeed A, Garcia-Losada P, Robins DA, Benson CT. Krishnan V, et al. Among authors: patel nj. Andrology. 2018 May;6(3):455-464. doi: 10.1111/andr.12479. Epub 2018 Mar 12. Andrology. 2018. PMID: 29527831 Free article. Clinical Trial.

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