Paquin JF - Search Results

1

Synthesis and biological evaluation of novel quinazoline-4-piperidinesulfamide derivatives as inhibitors of NPP1.

Forcellini E, Boutin S, Lefebvre CA, Shayhidin EE, Boulanger MC, Rhéaume G, Barbeau X, Lagüe P, Mathieu P, Paquin JF. Forcellini E, et al. Among authors: paquin jf. Eur J Med Chem. 2018 Mar 10;147:130-149. doi: 10.1016/j.ejmech.2018.01.094. Epub 2018 Feb 2. Eur J Med Chem. 2018. PMID: 29427906

2

Stereocontrolled approach to bromofluoroalkenes and their use for the synthesis of tri- and tetrasubstituted fluoroalkenes.

Landelle G, Champagne PA, Barbeau X, Paquin JF. Landelle G, et al. Among authors: paquin jf. Org Lett. 2009 Feb 5;11(3):681-4. doi: 10.1021/ol8027412. Org Lett. 2009. PMID: 19143558

3

Synthesis and growth inhibition activity of fluorinated derivatives of tamoxifen.

Malo-Forest B, Landelle G, Roy JA, Lacroix J, Gaudreault RC, Paquin JF. Malo-Forest B, et al. Among authors: paquin jf. Bioorg Med Chem Lett. 2013 Mar 15;23(6):1712-5. doi: 10.1016/j.bmcl.2013.01.057. Epub 2013 Jan 26. Bioorg Med Chem Lett. 2013. PMID: 23403084

4

Quinazoline-4-piperidine sulfamides are specific inhibitors of human NPP1 and prevent pathological mineralization of valve interstitial cells.

Shayhidin EE, Forcellini E, Boulanger MC, Mahmut A, Dautrey S, Barbeau X, Lagüe P, Sévigny J, Paquin JF, Mathieu P. Shayhidin EE, et al. Among authors: paquin jf. Br J Pharmacol. 2015 Aug;172(16):4189-99. doi: 10.1111/bph.13204. Epub 2015 Jul 8. Br J Pharmacol. 2015. PMID: 26031197 Free PMC article.

5

Synthesis of novel substituted pyrimidine derivatives bearing a sulfamide group and their in vitro cancer growth inhibition activity.

Lefebvre CA, Forcellini E, Boutin S, Côté MF, C-Gaudreault R, Mathieu P, Lagüe P, Paquin JF. Lefebvre CA, et al. Among authors: paquin jf. Bioorg Med Chem Lett. 2017 Jan 15;27(2):299-302. doi: 10.1016/j.bmcl.2016.11.052. Epub 2016 Nov 19. Bioorg Med Chem Lett. 2017. PMID: 27903409

6

Characterization of the structure, dynamics and allosteric pathways of human NPP1 in its free form and substrate-bound complex from molecular modeling.

Barbeau X, Mathieu P, Paquin JF, Lagüe P. Barbeau X, et al. Among authors: paquin jf. Mol Biosyst. 2017 May 30;13(6):1058-1069. doi: 10.1039/c7mb00095b. Mol Biosyst. 2017. PMID: 28474020

7

Design, synthesis and biological evaluation studies of novel small molecule ENPP1 inhibitors for cancer immunotherapy.

Gangar M, Goyal S, Raykar D, Khurana P, Martis AM, Goswami A, Ghoshal I, Patel KV, Nagare Y, Raikar S, Mukherjee A, Cyriac R, Paquin JF, Kulkarni A. Gangar M, et al. Among authors: paquin jf. Bioorg Chem. 2022 Feb;119:105549. doi: 10.1016/j.bioorg.2021.105549. Epub 2021 Dec 11. Bioorg Chem. 2022. PMID: 34929517

8

Stereoselective synthesis of both stereoisomers of β-fluorostyrene derivatives from a common intermediate.

Landelle G, Turcotte-Savard MO, Angers L, Paquin JF. Landelle G, et al. Among authors: paquin jf. Org Lett. 2011 Mar 18;13(6):1568-71. doi: 10.1021/ol200302h. Epub 2011 Feb 21. Org Lett. 2011. PMID: 21338081

9

Design, synthesis, and applications of potential substitutes of t-Bu-phosphinooxazoline in Pd-catalyzed asymmetric transformations and their use for the improvement of the enantioselectivity in the Pd-catalyzed allylation reaction of fluorinated allyl enol carbonates.

Bélanger É, Pouliot MF, Courtemanche MA, Paquin JF. Bélanger É, et al. Among authors: paquin jf. J Org Chem. 2012 Jan 6;77(1):317-31. doi: 10.1021/jo2019653. Epub 2011 Dec 7. J Org Chem. 2012. PMID: 22148548

10

Synthesis and properties of monofluorinated dimyristoylphosphatidylcholine derivatives: potential fluorinated probes for the study of membrane topology.

Guimond-Tremblay J, Gagnon MC, Pineault-Maltais JA, Turcotte V, Auger M, Paquin JF. Guimond-Tremblay J, et al. Among authors: paquin jf. Org Biomol Chem. 2012 Feb 14;10(6):1145-8. doi: 10.1039/c2ob06570c. Epub 2011 Dec 19. Org Biomol Chem. 2012. PMID: 22179779

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