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A vinylogous Norrish reaction as a strategy for light-mediated ring expansion.
Chem Commun (Camb). 2022 Feb 24;58(17):2910-2913. doi: 10.1039/d2cc00513a.
Chem Commun (Camb). 2022.
PMID: 35144274
Identification of ligand linkage vectors for the development of p300/CBP degraders.
Brownsey DK, Rowley BC, Gorobets E, Mihara K, Maity R, Papatzimas JW, Gelfand BS, Hollenberg MD, Bahlis NJ, Derksen DJ.
Brownsey DK, et al. Among authors: papatzimas jw.
RSC Med Chem. 2022 Apr 14;13(6):726-730. doi: 10.1039/d1md00070e. eCollection 2022 Jun 22.
RSC Med Chem. 2022.
PMID: 35814928
Free PMC article.
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From Inhibition to Degradation: Targeting the Antiapoptotic Protein Myeloid Cell Leukemia 1 (MCL1).
Papatzimas JW, Gorobets E, Maity R, Muniyat MI, MacCallum JL, Neri P, Bahlis NJ, Derksen DJ.
Papatzimas JW, et al.
J Med Chem. 2019 Jun 13;62(11):5522-5540. doi: 10.1021/acs.jmedchem.9b00455. Epub 2019 Jun 4.
J Med Chem. 2019.
PMID: 31117518
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ADAM protease inhibition overcomes resistance of breast cancer stem-like cells to γδ T cell immunotherapy.
Dutta I, Dieters-Castator D, Papatzimas JW, Medina A, Schueler J, Derksen DJ, Lajoie G, Postovit LM, Siegers GM.
Dutta I, et al. Among authors: papatzimas jw.
Cancer Lett. 2021 Jan 1;496:156-168. doi: 10.1016/j.canlet.2020.10.013. Epub 2020 Oct 10.
Cancer Lett. 2021.
PMID: 33045304
Free article.
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Correction to "Rational Chemical Design of Molecular Glue Degraders".
Toriki ES, Papatzimas JW, Nishikawa K, Dovala D, Frank AO, Hesse MJ, Dankova D, Song JG, Bruce-Smythe M, Struble H, Garcia FJ, Brittain SM, Kile AC, McGregor LM, McKenna JM, Tallarico JA, Schirle M, Nomura DK.
Toriki ES, et al. Among authors: papatzimas jw.
ACS Cent Sci. 2023 Jul 21;9(8):1702. doi: 10.1021/acscentsci.3c00844. eCollection 2023 Aug 23.
ACS Cent Sci. 2023.
PMID: 37637749
Free PMC article.
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Rational Chemical Design of Molecular Glue Degraders.
Toriki ES, Papatzimas JW, Nishikawa K, Dovala D, Frank AO, Hesse MJ, Dankova D, Song JG, Bruce-Smythe M, Struble H, Garcia FJ, Brittain SM, Kile AC, McGregor LM, McKenna JM, Tallarico JA, Schirle M, Nomura DK.
Toriki ES, et al. Among authors: papatzimas jw.
ACS Cent Sci. 2023 Apr 11;9(5):915-926. doi: 10.1021/acscentsci.2c01317. eCollection 2023 May 24.
ACS Cent Sci. 2023.
PMID: 37252349
Free PMC article.
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