Palmer BD - Search Results

1

Synthesis and Structure-Activity Relationships for the Anti-Mycobacterial Activity of 3-Phenyl-N-(Pyridin-2-ylmethyl)Pyrazolo[1,5-a]Pyrimidin-7-Amines.

Sutherland HS, Choi PJ, Lu GL, Giddens AC, Tong AST, Franzblau SG, Cooper CB, Palmer BD, Denny WA. Sutherland HS, et al. Among authors: palmer bd. Pharmaceuticals (Basel). 2022 Sep 8;15(9):1125. doi: 10.3390/ph15091125. Pharmaceuticals (Basel). 2022. PMID: 36145345 Free PMC article.

2

Synthetic Studies to Help Elucidate the Metabolism of the Preclinical Candidate TBAJ-876-A Less Toxic and More Potent Analogue of Bedaquiline.

Choi PJ, Conole D, Sutherland HS, Blaser A, Tong AST, Cooper CB, Upton AM, Palmer BD, Denny WA. Choi PJ, et al. Among authors: palmer bd. Molecules. 2020 Mar 20;25(6):1423. doi: 10.3390/molecules25061423. Molecules. 2020. PMID: 32245020 Free PMC article.

3

Synthesis and structure-activity relationships for tetrahydroisoquinoline-based inhibitors of Mycobacterium tuberculosis.

Lu GL, Tong AST, Conole D, Sutherland HS, Choi PJ, Franzblau SG, Upton AM, Lotlikar MU, Cooper CB, Denny WA, Palmer BD. Lu GL, et al. Among authors: palmer bd. Bioorg Med Chem. 2020 Nov 15;28(22):115784. doi: 10.1016/j.bmc.2020.115784. Epub 2020 Sep 24. Bioorg Med Chem. 2020. PMID: 33007562 Free PMC article.

4

Synthesis and structure-activity relationships for a new class of tetrahydronaphthalene amide inhibitors of Mycobacterium tuberculosis.

Sutherland HS, Lu GL, Tong AST, Conole D, Franzblau SG, Upton AM, Lotlikar MU, Cooper CB, Palmer BD, Choi PJ, Denny WA. Sutherland HS, et al. Among authors: palmer bd. Eur J Med Chem. 2022 Feb 5;229:114059. doi: 10.1016/j.ejmech.2021.114059. Epub 2021 Dec 21. Eur J Med Chem. 2022. PMID: 34963068 Free PMC article.

5

Synthetic studies towards isomeric pyrazolopyrimidines as potential ATP synthesis inhibitors of Mycobacterium tuberculosis. Structural correction of reported N-(6-(2-(dimethylamino)ethoxy)-5-fluoropyridin-3-yl)-2-(4-fluorophenyl)-5-(trifluoromethyl)pyrazolo[1,5-α]pyrimidin-7-amine.

Choi PJ, Lu GL, Sutherland HS, Giddens AC, Franzblau SG, Cooper CB, Denny WA, Palmer BD. Choi PJ, et al. Among authors: palmer bd. Tetrahedron Lett. 2022 Feb 2;90:None. doi: 10.1016/j.tetlet.2021.153611. Tetrahedron Lett. 2022. PMID: 35140452 Free PMC article.

6

Synthesis and structure-activity studies of biphenyl analogues of the tuberculosis drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824).

Palmer BD, Thompson AM, Sutherland HS, Blaser A, Kmentova I, Franzblau SG, Wan B, Wang Y, Ma Z, Denny WA. Palmer BD, et al. J Med Chem. 2010 Jan 14;53(1):282-94. doi: 10.1021/jm901207n. J Med Chem. 2010. PMID: 19928920

7

Synthesis and structure-activity relationships of antitubercular 2-nitroimidazooxazines bearing heterocyclic side chains.

Sutherland HS, Blaser A, Kmentova I, Franzblau SG, Wan B, Wang Y, Ma Z, Palmer BD, Denny WA, Thompson AM. Sutherland HS, et al. Among authors: palmer bd. J Med Chem. 2010 Jan 28;53(2):855-66. doi: 10.1021/jm901378u. J Med Chem. 2010. PMID: 19968290

8

Synthesis and structure-activity relationships of aza- and diazabiphenyl analogues of the antitubercular drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazine (PA-824).

Kmentova I, Sutherland HS, Palmer BD, Blaser A, Franzblau SG, Wan B, Wang Y, Ma Z, Denny WA, Thompson AM. Kmentova I, et al. Among authors: palmer bd. J Med Chem. 2010 Dec 9;53(23):8421-39. doi: 10.1021/jm101288t. Epub 2010 Nov 11. J Med Chem. 2010. PMID: 21069962

9

The nitroimidazooxazines (PA-824 and analogs): structure-activity relationship and mechanistic studies.

Denny WA, Palmer BD. Denny WA, et al. Among authors: palmer bd. Future Med Chem. 2010 Aug;2(8):1295-304. doi: 10.4155/fmc.10.207. Future Med Chem. 2010. PMID: 21426020 Review.

10

Synthesis and structure-activity relationships of varied ether linker analogues of the antitubercular drug (6S)-2-nitro-6-{[4-(trifluoromethoxy)benzyl]oxy}-6,7-dihydro-5h-imidazo[2,1-b][1,3]oxazine (PA-824).

Thompson AM, Sutherland HS, Palmer BD, Kmentova I, Blaser A, Franzblau SG, Wan B, Wang Y, Ma Z, Denny WA. Thompson AM, et al. Among authors: palmer bd. J Med Chem. 2011 Oct 13;54(19):6563-85. doi: 10.1021/jm200377r. Epub 2011 Sep 1. J Med Chem. 2011. PMID: 21846109

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