Pace S - Search Results

1

Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E₂ and Leukotriene Biosynthesis Inhibitors.

Potenza M, Giordano A, Chini MG, Saviano A, Kretzer C, Raucci F, Russo M, Lauro G, Terracciano S, Bruno I, Iorizzi M, Hofstetter RK, Pace S, Maione F, Werz O, Bifulco G. Potenza M, et al. Among authors: pace s. ACS Med Chem Lett. 2022 Dec 9;14(1):26-34. doi: 10.1021/acsmedchemlett.2c00343. eCollection 2023 Jan 12. ACS Med Chem Lett. 2022. PMID: 36655121 Free PMC article.

2

The novel benzimidazole derivative BRP-7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5-lipoxygenase-activating protein (FLAP).

Pergola C, Gerstmeier J, Mönch B, Çalışkan B, Luderer S, Weinigel C, Barz D, Maczewsky J, Pace S, Rossi A, Sautebin L, Banoglu E, Werz O. Pergola C, et al. Among authors: pace s. Br J Pharmacol. 2014 Jun;171(12):3051-64. doi: 10.1111/bph.12625. Br J Pharmacol. 2014. PMID: 24641614 Free PMC article.

3

In vivo sex differences in leukotriene biosynthesis in zymosan-induced peritonitis.

Rossi A, Pergola C, Pace S, Rådmark O, Werz O, Sautebin L. Rossi A, et al. Among authors: pace s. Pharmacol Res. 2014 Sep;87:1-7. doi: 10.1016/j.phrs.2014.05.011. Epub 2014 Jun 2. Pharmacol Res. 2014. PMID: 24892983

4

SAR studies on curcumin's pro-inflammatory targets: discovery of prenylated pyrazolocurcuminoids as potent and selective novel inhibitors of 5-lipoxygenase.

Koeberle A, Muñoz E, Appendino GB, Minassi A, Pace S, Rossi A, Weinigel C, Barz D, Sautebin L, Caprioglio D, Collado JA, Werz O. Koeberle A, et al. Among authors: pace s. J Med Chem. 2014 Jul 10;57(13):5638-48. doi: 10.1021/jm500308c. Epub 2014 Jun 24. J Med Chem. 2014. PMID: 24920381

5

The hallucinogenic diterpene salvinorin A inhibits leukotriene synthesis in experimental models of inflammation.

Rossi A, Pace S, Tedesco F, Pagano E, Guerra G, Troisi F, Werner M, Roviezzo F, Zjawiony JK, Werz O, Izzo AA, Capasso R. Rossi A, et al. Among authors: pace s. Pharmacol Res. 2016 Apr;106:64-71. doi: 10.1016/j.phrs.2016.01.032. Epub 2016 Feb 6. Pharmacol Res. 2016. PMID: 26859523

6

Humudifucol and Bioactive Prenylated Polyphenols from Hops (Humulus lupulus cv. "Cascade").

Forino M, Pace S, Chianese G, Santagostini L, Werner M, Weinigel C, Rummler S, Fico G, Werz O, Taglialatela-Scafati O. Forino M, et al. Among authors: pace s. J Nat Prod. 2016 Mar 25;79(3):590-7. doi: 10.1021/acs.jnatprod.5b01052. Epub 2016 Feb 26. J Nat Prod. 2016. PMID: 26918635

7

The 5-lipoxygenase inhibitor RF-22c potently suppresses leukotriene biosynthesis in cellulo and blocks bronchoconstriction and inflammation in vivo.

Schaible AM, Filosa R, Krauth V, Temml V, Pace S, Garscha U, Liening S, Weinigel C, Rummler S, Schieferdecker S, Nett M, Peduto A, Collarile S, Scuotto M, Roviezzo F, Spaziano G, de Rosa M, Stuppner H, Schuster D, D'Agostino B, Werz O. Schaible AM, et al. Among authors: pace s. Biochem Pharmacol. 2016 Jul 15;112:60-71. doi: 10.1016/j.bcp.2016.04.019. Epub 2016 May 5. Biochem Pharmacol. 2016. PMID: 27157409

8

Anti-inflammatory and analgesic activity of carnosol and carnosic acid in vivo and in vitro and in silico analysis of their target interactions.

Maione F, Cantone V, Pace S, Chini MG, Bisio A, Romussi G, Pieretti S, Werz O, Koeberle A, Mascolo N, Bifulco G. Maione F, et al. Among authors: pace s. Br J Pharmacol. 2017 Jun;174(11):1497-1508. doi: 10.1111/bph.13545. Epub 2016 Aug 8. Br J Pharmacol. 2017. PMID: 27464306 Free PMC article.

9

BRP-187: A potent inhibitor of leukotriene biosynthesis that acts through impeding the dynamic 5-lipoxygenase/5-lipoxygenase-activating protein (FLAP) complex assembly.

Garscha U, Voelker S, Pace S, Gerstmeier J, Emini B, Liening S, Rossi A, Weinigel C, Rummler S, Schubert US, Scriba GK, Çelikoğlu E, Çalışkan B, Banoglu E, Sautebin L, Werz O. Garscha U, et al. Among authors: pace s. Biochem Pharmacol. 2016 Nov 1;119:17-26. doi: 10.1016/j.bcp.2016.08.023. Epub 2016 Aug 31. Biochem Pharmacol. 2016. PMID: 27592027

10

Myxochelin-Inspired 5-Lipoxygenase Inhibitors: Synthesis and Biological Evaluation.

Schieferdecker S, König S, Pace S, Werz O, Nett M. Schieferdecker S, et al. Among authors: pace s. ChemMedChem. 2017 Jan 5;12(1):23-27. doi: 10.1002/cmdc.201600536. Epub 2016 Nov 29. ChemMedChem. 2017. PMID: 27875023

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