Overkleeft HS - Search Results

1

Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition.

Ogasawara D, Deng H, Viader A, Baggelaar MP, Breman A, den Dulk H, van den Nieuwendijk AM, Soethoudt M, van der Wel T, Zhou J, Overkleeft HS, Sanchez-Alavez M, Mori S, Nguyen W, Conti B, Liu X, Chen Y, Liu QS, Cravatt BF, van der Stelt M. Ogasawara D, et al. Among authors: overkleeft hs. Proc Natl Acad Sci U S A. 2016 Jan 5;113(1):26-33. doi: 10.1073/pnas.1522364112. Epub 2015 Dec 14. Proc Natl Acad Sci U S A. 2016. PMID: 26668358 Free PMC article.

2

Extending solid-phase methods in inorganic synthesis: the first dinuclear platinum complex synthesised via the solid phase.

van Zutphen S, Robillard MS, van der Marel GA, Overkleeft HS, den Dulk H, Brouwer J, Reedijk J. van Zutphen S, et al. Among authors: overkleeft hs. Chem Commun (Camb). 2003 Mar 7;(5):634-5. doi: 10.1039/b212388f. Chem Commun (Camb). 2003. PMID: 12669861

3

Development of an isotope-coded activity-based probe for the quantitative profiling of cysteine proteases.

van Swieten PF, Maehr R, van den Nieuwendijk AM, Kessler BM, Reich M, Wong CS, Kalbacher H, Leeuwenburgh MA, Driessen C, van der Marel GA, Ploegh HL, Overkleeft HS. van Swieten PF, et al. Among authors: overkleeft hs. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3131-4. doi: 10.1016/j.bmcl.2004.04.046. Bioorg Med Chem Lett. 2004. PMID: 15149659

4

Combinatorial discovery of new asymmetric cis platinum anticancer complexes is made possible with solid-phase synthetic methods.

van Zutphen S, Stone EA, van Rijt S, Robillard MS, van der Marel GA, Overkleeft HS, den Dulk H, Brouwer J, Reedijk J. van Zutphen S, et al. Among authors: overkleeft hs. J Inorg Biochem. 2005 Oct;99(10):2032-8. doi: 10.1016/j.jinorgbio.2005.06.033. J Inorg Biochem. 2005. PMID: 16099049

5

A fluorescent broad-spectrum proteasome inhibitor for labeling proteasomes in vitro and in vivo.

Verdoes M, Florea BI, Menendez-Benito V, Maynard CJ, Witte MD, van der Linden WA, van den Nieuwendijk AM, Hofmann T, Berkers CR, van Leeuwen FW, Groothuis TA, Leeuwenburgh MA, Ovaa H, Neefjes JJ, Filippov DV, van der Marel GA, Dantuma NP, Overkleeft HS. Verdoes M, et al. Among authors: overkleeft hs. Chem Biol. 2006 Nov;13(11):1217-26. doi: 10.1016/j.chembiol.2006.09.013. Chem Biol. 2006. PMID: 17114003

6

A cell-permeable inhibitor and activity-based probe for the caspase-like activity of the proteasome.

van Swieten PF, Samuel E, Hernández RO, van den Nieuwendijk AM, Leeuwenburgh MA, van der Marel GA, Kessler BM, Overkleeft HS, Kisselev AF. van Swieten PF, et al. Among authors: overkleeft hs. Bioorg Med Chem Lett. 2007 Jun 15;17(12):3402-5. doi: 10.1016/j.bmcl.2007.03.092. Epub 2007 Apr 2. Bioorg Med Chem Lett. 2007. PMID: 17442566

7

Mixing of peptides and electrophilic traps gives rise to potent, broad-spectrum proteasome inhibitors.

Verdoes M, Florea BI, van der Linden WA, Renou D, van den Nieuwendijk AM, van der Marel GA, Overkleeft HS. Verdoes M, et al. Among authors: overkleeft hs. Org Biomol Chem. 2007 May 7;5(9):1416-26. doi: 10.1039/b702268a. Epub 2007 Mar 23. Org Biomol Chem. 2007. PMID: 17464411

8

Incorporation of fluorinated phenylalanine generates highly specific inhibitor of proteasome's chymotrypsin-like sites.

Geurink PP, Liu N, Spaans MP, Downey SL, van den Nieuwendijk AM, van der Marel GA, Kisselev AF, Florea BI, Overkleeft HS. Geurink PP, et al. Among authors: overkleeft hs. J Med Chem. 2010 Mar 11;53(5):2319-23. doi: 10.1021/jm9015685. J Med Chem. 2010. PMID: 20131905 Free PMC article.

9

Synthesis of L-altro-1-deoxynojirimycin, D-allo-1-deoxynojirimycin, and D-galacto-1-deoxynojirimycin from a single chiral cyanohydrin.

van den Nieuwendijk AM, Ruben M, Engelsma SE, Risseeuw MD, van den Berg RJ, Boot RG, Aerts JM, Brussee J, van der Marel GA, Overkleeft HS. van den Nieuwendijk AM, et al. Among authors: overkleeft hs. Org Lett. 2010 Sep 3;12(17):3957-9. doi: 10.1021/ol101556k. Org Lett. 2010. PMID: 20690611

10

Activity-based profiling reveals reactivity of the murine thymoproteasome-specific subunit beta5t.

Florea BI, Verdoes M, Li N, van der Linden WA, Geurink PP, van den Elst H, Hofmann T, de Ru A, van Veelen PA, Tanaka K, Sasaki K, Murata S, den Dulk H, Brouwer J, Ossendorp FA, Kisselev AF, Overkleeft HS. Florea BI, et al. Among authors: overkleeft hs. Chem Biol. 2010 Aug 27;17(8):795-801. doi: 10.1016/j.chembiol.2010.05.027. Chem Biol. 2010. PMID: 20797608 Free PMC article.

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