Overkleeft HS - Search Results

1

Activity-based profiling reveals reactivity of the murine thymoproteasome-specific subunit beta5t.

Florea BI, Verdoes M, Li N, van der Linden WA, Geurink PP, van den Elst H, Hofmann T, de Ru A, van Veelen PA, Tanaka K, Sasaki K, Murata S, den Dulk H, Brouwer J, Ossendorp FA, Kisselev AF, Overkleeft HS. Florea BI, et al. Among authors: overkleeft hs. Chem Biol. 2010 Aug 27;17(8):795-801. doi: 10.1016/j.chembiol.2010.05.027. Chem Biol. 2010. PMID: 20797608 Free PMC article.

2

Extended peptide-based inhibitors efficiently target the proteasome and reveal overlapping specificities of the catalytic beta-subunits.

Kessler BM, Tortorella D, Altun M, Kisselev AF, Fiebiger E, Hekking BG, Ploegh HL, Overkleeft HS. Kessler BM, et al. Among authors: overkleeft hs. Chem Biol. 2001 Sep;8(9):913-29. doi: 10.1016/s1074-5521(01)00069-2. Chem Biol. 2001. PMID: 11564559

3

Extending solid-phase methods in inorganic synthesis: the first dinuclear platinum complex synthesised via the solid phase.

van Zutphen S, Robillard MS, van der Marel GA, Overkleeft HS, den Dulk H, Brouwer J, Reedijk J. van Zutphen S, et al. Among authors: overkleeft hs. Chem Commun (Camb). 2003 Mar 7;(5):634-5. doi: 10.1039/b212388f. Chem Commun (Camb). 2003. PMID: 12669861

4

The caspase-like sites of proteasomes, their substrate specificity, new inhibitors and substrates, and allosteric interactions with the trypsin-like sites.

Kisselev AF, Garcia-Calvo M, Overkleeft HS, Peterson E, Pennington MW, Ploegh HL, Thornberry NA, Goldberg AL. Kisselev AF, et al. Among authors: overkleeft hs. J Biol Chem. 2003 Sep 19;278(38):35869-77. doi: 10.1074/jbc.M303725200. Epub 2003 Jun 18. J Biol Chem. 2003. PMID: 12815064 Free article.

5

The use of a mannitol-derived fused oxacycle as a combinatorial scaffold.

Timmer MS, Verdoes M, Sliedregt LA, van der Marel GA, van Boom JH, Overkleeft HS. Timmer MS, et al. Among authors: overkleeft hs. J Org Chem. 2003 Nov 28;68(24):9406-11. doi: 10.1021/jo0349429. J Org Chem. 2003. PMID: 14629165

6

An unusual reverse turn structure adopted by a furanoid sugar amino acid incorporated in gramicidin S.

Grotenbreg GM, Timmer MS, Llamas-Saiz AL, Verdoes M, van der Marel GA, van Raaij MJ, Overkleeft HS, Overhand M. Grotenbreg GM, et al. Among authors: overkleeft hs. J Am Chem Soc. 2004 Mar 24;126(11):3444-6. doi: 10.1021/ja0397254. J Am Chem Soc. 2004. PMID: 15025470

7

Development of an isotope-coded activity-based probe for the quantitative profiling of cysteine proteases.

van Swieten PF, Maehr R, van den Nieuwendijk AM, Kessler BM, Reich M, Wong CS, Kalbacher H, Leeuwenburgh MA, Driessen C, van der Marel GA, Ploegh HL, Overkleeft HS. van Swieten PF, et al. Among authors: overkleeft hs. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3131-4. doi: 10.1016/j.bmcl.2004.04.046. Bioorg Med Chem Lett. 2004. PMID: 15149659

8

Design, synthesis, and evaluation of sugar amino acid based inhibitors of protein prenyl transferases PFT and PGGT-1.

El Oualid F, Burm BE, Leroy IM, Cohen LH, van Boom JH, van den Elst H, Overkleeft HS, van der Marel GA, Overhand M. El Oualid F, et al. Among authors: overkleeft hs. J Med Chem. 2004 Jul 29;47(16):3920-3. doi: 10.1021/jm049927q. J Med Chem. 2004. PMID: 15267228

9

A practical synthesis of gramicidin s and sugar amino Acid containing analogues.

Grotenbreg GM, Kronemeijer M, Timmer MS, El Oualid F, van Well RM, Verdoes M, Spalburg E, van Hooft PA, de Neeling AJ, Noort D, van Boom JH, van der Marel GA, Overkleeft HS, Overhand M. Grotenbreg GM, et al. Among authors: overkleeft hs. J Org Chem. 2004 Nov 12;69(23):7851-9. doi: 10.1021/jo0487449. J Org Chem. 2004. PMID: 15527261

10

Synthesis and biological evaluation of lipophilic Ca(1)a(2)L analogues as potential bisubstrate inhibitors of protein:geranylgeranyl transferase-1.

El Oualid F, Baktawar J, Leroy IM, van den Elst H, Cohen LH, van der Marel GA, Overkleeft HS, Overhand M. El Oualid F, et al. Among authors: overkleeft hs. Bioorg Med Chem. 2005 Mar 1;13(5):1463-75. doi: 10.1016/j.bmc.2004.12.035. Bioorg Med Chem. 2005. PMID: 15698762

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