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Recent approaches to chemical discovery and development against malaria and the neglected tropical diseases human African trypanosomiasis and schistosomiasis.
Chem Rev. 2014 Nov 26;114(22):11138-63. doi: 10.1021/cr500098f. Epub 2014 Jul 11.
Chem Rev. 2014.
PMID: 25014712
Review.
No abstract available.
Artemisinin derivatives: a patent review (2006 - present).
Njuguna NM, Ongarora DS, Chibale K.
Njuguna NM, et al.
Expert Opin Ther Pat. 2012 Oct;22(10):1179-203. doi: 10.1517/13543776.2012.724063. Epub 2012 Sep 13.
Expert Opin Ther Pat. 2012.
PMID: 22971128
Review.
Item in Clipboard
Identification and characterization of reactive metabolites in natural products-driven drug discovery.
Njuguna NM, Masimirembwa C, Chibale K.
Njuguna NM, et al.
J Nat Prod. 2012 Mar 23;75(3):507-13. doi: 10.1021/np200786j. Epub 2012 Feb 1.
J Nat Prod. 2012.
PMID: 22296642
Review.
Item in Clipboard
In silico comparison of antimycobacterial natural products with known antituberculosis drugs.
Espinoza-Moraga M, Njuguna NM, Mugumbate G, Caballero J, Chibale K.
Espinoza-Moraga M, et al. Among authors: njuguna nm.
J Chem Inf Model. 2013 Mar 25;53(3):649-60. doi: 10.1021/ci300467b. Epub 2013 Feb 22.
J Chem Inf Model. 2013.
PMID: 23410241
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Chloroquine-containing compounds: a patent review (2010 - 2014).
Njaria PM, Okombo J, Njuguna NM, Chibale K.
Njaria PM, et al. Among authors: njuguna nm.
Expert Opin Ther Pat. 2015;25(9):1003-24. doi: 10.1517/13543776.2015.1050791. Epub 2015 Jun 1.
Expert Opin Ther Pat. 2015.
PMID: 26013494
Free PMC article.
Review.
Item in Clipboard
Improvement of the chemical inhibition phenotyping assay by cross-reactivity correction.
Njuguna NM, Umehara KI, Huth F, Schiller H, Chibale K, Camenisch G.
Njuguna NM, et al.
Drug Metab Pers Ther. 2016 Dec 1;31(4):221-228. doi: 10.1515/dmpt-2016-0028.
Drug Metab Pers Ther. 2016.
PMID: 27718490
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Meloxicam emulgels for topical management of rheumatism: Formulation development, in vitro and in vivo characterization.
Mwangi AN, Njogu PM, Maru SM, Njuguna NM, Njaria PM, Kiriiri GK, Mathenge AW.
Mwangi AN, et al. Among authors: njuguna nm.
Saudi Pharm J. 2021 Apr;29(4):351-360. doi: 10.1016/j.jsps.2021.03.005. Epub 2021 Mar 23.
Saudi Pharm J. 2021.
PMID: 33994830
Free PMC article.
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