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PI(18:1/18:1) is a SCD1-derived lipokine that limits stress signaling.
Nat Commun. 2022 May 27;13(1):2982. doi: 10.1038/s41467-022-30374-9.
Nat Commun. 2022.
PMID: 35624087
Free PMC article.
Endogenous metabolites of vitamin E limit inflammation by targeting 5-lipoxygenase.
Pein H, Ville A, Pace S, Temml V, Garscha U, Raasch M, Alsabil K, Viault G, Dinh CP, Guilet D, Troisi F, Neukirch K, König S, Bilancia R, Waltenberger B, Stuppner H, Wallert M, Lorkowski S, Weinigel C, Rummler S, Birringer M, Roviezzo F, Sautebin L, Helesbeux JJ, Séraphin D, Mosig AS, Schuster D, Rossi A, Richomme P, Werz O, Koeberle A.
Pein H, et al. Among authors: neukirch k.
Nat Commun. 2018 Sep 20;9(1):3834. doi: 10.1038/s41467-018-06158-5.
Nat Commun. 2018.
PMID: 30237488
Free PMC article.
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Exploration of Long-Chain Vitamin E Metabolites for the Discovery of a Highly Potent, Orally Effective, and Metabolically Stable 5-LOX Inhibitor that Limits Inflammation.
Neukirch K, Alsabil K, Dinh CP, Bilancia R, Raasch M, Ville A, Cerqua I, Viault G, Bréard D, Pace S, Temml V, Brunner E, Jordan PM, Marques MC, Loeser K, Gollowitzer A, Permann S, Gerstmeier J, Lorkowski S, Stuppner H, Garscha U, Rodrigues T, Bernardes GJL, Schuster D, Séraphin D, Richomme P, Rossi A, Mosig AS, Roviezzo F, Werz O, Helesbeux JJ, Koeberle A.
Neukirch K, et al.
J Med Chem. 2021 Aug 12;64(15):11496-11526. doi: 10.1021/acs.jmedchem.1c00806. Epub 2021 Jul 19.
J Med Chem. 2021.
PMID: 34279935
Free PMC article.
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Structure-based design, semi-synthesis and anti-inflammatory activity of tocotrienolic amides as 5-lipoxygenase inhibitors.
Dinh CP, Ville A, Neukirch K, Viault G, Temml V, Koeberle A, Werz O, Schuster D, Stuppner H, Richomme P, Helesbeux JJ, Séraphin D.
Dinh CP, et al. Among authors: neukirch k.
Eur J Med Chem. 2020 Sep 15;202:112518. doi: 10.1016/j.ejmech.2020.112518. Epub 2020 Jun 27.
Eur J Med Chem. 2020.
PMID: 32668380
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Learning from Nature: From a Marine Natural Product to Synthetic Cyclooxygenase-1 Inhibitors by Automated De Novo Design.
Friedrich L, Cingolani G, Ko YH, Iaselli M, Miciaccia M, Perrone MG, Neukirch K, Bobinger V, Merk D, Hofstetter RK, Werz O, Koeberle A, Scilimati A, Schneider G.
Friedrich L, et al. Among authors: neukirch k.
Adv Sci (Weinh). 2021 Aug;8(16):e2100832. doi: 10.1002/advs.202100832. Epub 2021 Jun 27.
Adv Sci (Weinh). 2021.
PMID: 34176236
Free PMC article.
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A vitamin E long-chain metabolite and the inspired drug candidate α-amplexichromanol relieve asthma features in an experimental model of allergen sensitization.
Cerqua I, Neukirch K, Terlizzi M, Granato E, Caiazzo E, Cicala C, Ialenti A, Capasso R, Werz O, Sorrentino R, Seraphin D, Helesbeux JJ, Cirino G, Koeberle A, Roviezzo F, Rossi A.
Cerqua I, et al. Among authors: neukirch k.
Pharmacol Res. 2022 Jul;181:106250. doi: 10.1016/j.phrs.2022.106250. Epub 2022 May 10.
Pharmacol Res. 2022.
PMID: 35562015
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Early age of onset in fatal familial insomnia. Two novel cases and review of the literature.
Harder A, Gregor A, Wirth T, Kreuz F, Schulz-Schaeffer WJ, Windl O, Plotkin M, Amthauer H, Neukirch K, Kretzschmar HA, Kuhlmann T, Braas R, Hahne HH, Jendroska K.
Harder A, et al. Among authors: neukirch k.
J Neurol. 2004 Jun;251(6):715-24. doi: 10.1007/s00415-004-0409-0.
J Neurol. 2004.
PMID: 15311348
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Computer aided planning device for preoperative bending of osteosynthesis plates.
Burghart CR, Neukirch K, Hassfeld S, Rembold U, Woern H.
Burghart CR, et al. Among authors: neukirch k.
Stud Health Technol Inform. 2000;70:46-52.
Stud Health Technol Inform. 2000.
PMID: 10977582
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