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Novel thienopyrimidones targeting hepatic and erythrocytic stages of Plasmodium parasites with increased microsomal stability.
Lagardère P, Mustière R, Amanzougaghene N, Hutter S, Casanova M, Franetich JF, Tajeri S, Malzert-Fréon A, Corvaisier S, Since M, Azas N, Vanelle P, Verhaeghe P, Primas N, Mazier D, Masurier N, Lisowski V. Lagardère P, et al. Among authors: mustiere r. Eur J Med Chem. 2023 Dec 5;261:115873. doi: 10.1016/j.ejmech.2023.115873. Epub 2023 Oct 13. Eur J Med Chem. 2023. PMID: 37857143
New antiplasmodial 4-amino-thieno[3,2-d]pyrimidines with improved intestinal permeability and microsomal stability.
Lagardère P, Mustière R, Amanzougaghene N, Hutter S, Casanova M, Franetich JF, Tajeri S, Malzert-Fréon A, Corvaisier S, Azas N, Vanelle P, Verhaeghe P, Primas N, Mazier D, Masurier N, Lisowski V. Lagardère P, et al. Among authors: mustiere r. Eur J Med Chem. 2023 Mar 5;249:115115. doi: 10.1016/j.ejmech.2023.115115. Epub 2023 Jan 13. Eur J Med Chem. 2023. PMID: 36680984
4-Substituted Thieno[3,2-d]pyrimidines as Dual-Stage Antiplasmodial Derivatives.
Lagardère P, Mustière R, Amanzougaghene N, Hutter S, Franetich JF, Azas N, Vanelle P, Verhaeghe P, Primas N, Mazier D, Masurier N, Lisowski V. Lagardère P, et al. Among authors: mustiere r. Pharmaceuticals (Basel). 2022 Jul 1;15(7):820. doi: 10.3390/ph15070820. Pharmaceuticals (Basel). 2022. PMID: 35890119 Free PMC article.
Synthesis of antiplasmodial 2-aminothieno[3,2-d]pyrimidin-4(3H)-one analogues using the scaffold hopping strategy.
Mustière R, Lagardère P, Hutter S, Dell'Orco V, Amanzougaghene N, Tajeri S, Franetich JF, Corvaisier S, Since M, Malzert-Fréon A, Masurier N, Lisowski V, Verhaeghe P, Mazier D, Azas N, Vanelle P, Primas N. Mustière R, et al. Eur J Med Chem. 2022 Nov 5;241:114619. doi: 10.1016/j.ejmech.2022.114619. Epub 2022 Jul 20. Eur J Med Chem. 2022. PMID: 35872545
A New Thienopyrimidinone Chemotype Shows Multistage Activity against Plasmodium falciparum, Including Artemisinin-Resistant Parasites.
Bosson-Vanga H, Primas N, Franetich JF, Lavazec C, Gomez L, Ashraf K, Tefit M, Soulard V, Dereuddre-Bosquet N, Le Grand R, Donnette M, Mustière R, Amanzougaghene N, Tajeri S, Suzanne P, Malzert-Fréon A, Rault S, Vanelle P, Hutter S, Cohen A, Snounou G, Roques P, Azas N, Lagardère P, Lisowski V, Masurier N, Nguyen M, Paloque L, Benoit-Vical F, Verhaeghe P, Mazier D. Bosson-Vanga H, et al. Among authors: mustiere r. Microbiol Spectr. 2021 Oct 31;9(2):e0027421. doi: 10.1128/Spectrum.00274-21. Epub 2021 Sep 29. Microbiol Spectr. 2021. PMID: 34724729 Free PMC article.