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An insight into the anticancer potential of carbamates and thiocarbamates of 10-demethoxy-10-methylaminocolchicine.
Eur J Med Chem. 2021 Apr 5;215:113282. doi: 10.1016/j.ejmech.2021.113282. Epub 2021 Feb 10.
Eur J Med Chem. 2021.
PMID: 33611191
Free article.
Synthesis, Antiproliferative Activity and Molecular Docking Studies of Novel Doubly Modified Colchicine Amides and Sulfonamides as Anticancer Agents.
Krzywik J, Mozga W, Aminpour M, Janczak J, Maj E, Wietrzyk J, Tuszyński JA, Huczyński A.
Krzywik J, et al. Among authors: mozga w.
Molecules. 2020 Apr 14;25(8):1789. doi: 10.3390/molecules25081789.
Molecules. 2020.
PMID: 32295119
Free PMC article.
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New Series of Double-Modified Colchicine Derivatives: Synthesis, Cytotoxic Effect and Molecular Docking.
Krzywik J, Aminpour M, Maj E, Mozga W, Wietrzyk J, Tuszyński JA, Huczyński A.
Krzywik J, et al. Among authors: mozga w.
Molecules. 2020 Aug 2;25(15):3540. doi: 10.3390/molecules25153540.
Molecules. 2020.
PMID: 32748887
Free PMC article.
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Synthesis and antiproliferative screening of novel doubly modified colchicines containing urea, thiourea and guanidine moieties.
Krzywik J, Maj E, Nasulewicz-Goldeman A, Mozga W, Wietrzyk J, Huczyński A.
Krzywik J, et al. Among authors: mozga w.
Bioorg Med Chem Lett. 2021 Sep 1;47:128197. doi: 10.1016/j.bmcl.2021.128197. Epub 2021 Jun 8.
Bioorg Med Chem Lett. 2021.
PMID: 34116158
Free article.
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Novel Double-Modified Colchicine Derivatives Bearing 1,2,3-Triazole: Design, Synthesis, and Biological Activity Evaluation.
Krzywik J, Nasulewicz-Goldeman A, Mozga W, Wietrzyk J, Huczyński A.
Krzywik J, et al. Among authors: mozga w.
ACS Omega. 2021 Sep 28;6(40):26583-26600. doi: 10.1021/acsomega.1c03948. eCollection 2021 Oct 12.
ACS Omega. 2021.
PMID: 34661013
Free PMC article.
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Discovery of OATD-01, a First-in-Class Chitinase Inhibitor as Potential New Therapeutics for Idiopathic Pulmonary Fibrosis.
Koralewski R, Dymek B, Mazur M, Sklepkiewicz P, Olejniczak S, Czestkowski W, Matyszewski K, Andryianau G, Niedziejko P, Kowalski M, Gruza M, Borek B, Jedrzejczak K, Bartoszewicz A, Pluta E, Rymaszewska A, Kania M, Rejczak T, Piasecka S, Mlacki M, Mazurkiewicz M, Piotrowicz M, Salamon M, Zagozdzon A, Napiorkowska-Gromadzka A, Bartlomiejczak A, Mozga W, Dobrzański P, Dzwonek K, Golab J, Nowotny M, Olczak J, Golebiowski A.
Koralewski R, et al. Among authors: mozga w.
J Med Chem. 2020 Dec 24;63(24):15527-15540. doi: 10.1021/acs.jmedchem.0c01179. Epub 2020 Oct 20.
J Med Chem. 2020.
PMID: 33078933
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Development of Dual Chitinase Inhibitors as Potential New Treatment for Respiratory System Diseases.
Mazur M, Dymek B, Koralewski R, Sklepkiewicz P, Olejniczak S, Mazurkiewicz M, Piotrowicz M, Salamon M, Jędrzejczak K, Zagozdzon A, Czestkowski W, Matyszewski K, Borek B, Bartoszewicz A, Pluta E, Rymaszewska A, Mozga W, Stefaniak F, Dobrzański P, Dzwonek K, Golab J, Golebiowski A, Olczak J.
Mazur M, et al. Among authors: mozga w.
J Med Chem. 2019 Aug 8;62(15):7126-7145. doi: 10.1021/acs.jmedchem.9b00681. Epub 2019 Jul 23.
J Med Chem. 2019.
PMID: 31291098
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Solution conformational study of Scyliorhinin I analogues with conformational constraints by two-dimensional NMR and theoretical conformational analysis.
Rodziewicz-Motowidło S, Legowska A, Qi XF, Czaplewski C, Liwo A, Sowiński P, Mozga W, Olczak J, Zabrocki J, Rolka K.
Rodziewicz-Motowidło S, et al. Among authors: mozga w.
J Pept Res. 2000 Sep;56(3):132-46. doi: 10.1034/j.1399-3011.2000.00697.x.
J Pept Res. 2000.
PMID: 11007270
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