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Do Small Molecules Activate the TrkB Receptor in the Same Manner as BDNF? Limitations of Published TrkB Low Molecular Agonists and Screening for Novel TrkB Orthosteric Agonists.
Pharmaceuticals (Basel). 2021 Jul 21;14(8):704. doi: 10.3390/ph14080704.
Pharmaceuticals (Basel). 2021.
PMID: 34451801
Free PMC article.
Esketamine inhaled as dry powder: Pharmacokinetic, pharmacodynamic and safety assessment in a preclinical study.
Matłoka M, Janowska S, Gajos-Draus A, Ziółkowski H, Janicka M, Perko P, Kamil K, Pankiewicz P, Moszczyński-Pętkowski R, Mach M, Dera P, Abramski K, Teska-Kamińska M, Tratkiewicz E, Wieczorek M, Pieczykolan J.
Matłoka M, et al. Among authors: moszczynski petkowski r.
Pulm Pharmacol Ther. 2022 Jun;73-74:102127. doi: 10.1016/j.pupt.2022.102127. Epub 2022 Apr 14.
Pulm Pharmacol Ther. 2022.
PMID: 35429651
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Synthesis and characterization of novel classes of PDE10A inhibitors - 1H-1,3-benzodiazoles and imidazo[1,2-a]pyrimidines.
Moszczyński-Pętkowski R, Majer J, Borkowska M, Bojarski Ł, Janowska S, Matłoka M, Stefaniak F, Smuga D, Bazydło K, Dubiel K, Wieczorek M.
Moszczyński-Pętkowski R, et al.
Eur J Med Chem. 2018 Jul 15;155:96-116. doi: 10.1016/j.ejmech.2018.05.043. Epub 2018 May 30.
Eur J Med Chem. 2018.
PMID: 29870883
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Virtual screening-driven discovery of dual 5-HT6/5-HT2A receptor ligands with pro-cognitive properties.
Staroń J, Kurczab R, Warszycki D, Satała G, Krawczyk M, Bugno R, Lenda T, Popik P, Hogendorf AS, Hogendorf A, Dubiel K, Matłoka M, Moszczyński-Pętkowski R, Pieczykolan J, Wieczorek M, Zajdel P, Bojarski AJ.
Staroń J, et al. Among authors: moszczynski petkowski r.
Eur J Med Chem. 2020 Jan 1;185:111857. doi: 10.1016/j.ejmech.2019.111857. Epub 2019 Nov 7.
Eur J Med Chem. 2020.
PMID: 31734022
Free article.
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Pyrroloquinoline scaffold-based 5-HT6R ligands: Synthesis, quantum chemical and molecular dynamic studies, and influence of nitrogen atom position in the scaffold on affinity.
Grychowska K, Kurczab R, Śliwa P, Satała G, Dubiel K, Matłoka M, Moszczyński-Pętkowski R, Pieczykolan J, Bojarski AJ, Zajdel P.
Grychowska K, et al. Among authors: moszczynski petkowski r.
Bioorg Med Chem. 2018 Jul 23;26(12):3588-3595. doi: 10.1016/j.bmc.2018.05.033. Epub 2018 May 23.
Bioorg Med Chem. 2018.
PMID: 29853337
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Quetiapine and novel PDE10A inhibitors potentiate the anti-BuChE activity of donepezil.
Sikora J, Podsiedlik M, Pietras T, Kosmalski M, Matłoka M, Moszczyński-Petkowski R, Wieczorek M, Markowicz-Piasecka M.
Sikora J, et al. Among authors: moszczynski petkowski r.
J Enzyme Inhib Med Chem. 2020 Dec;35(1):1743-1750. doi: 10.1080/14756366.2020.1818739.
J Enzyme Inhib Med Chem. 2020.
PMID: 32938236
Free PMC article.
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2-Aminoimidazole-based antagonists of the 5-HT6 receptor - A new concept in aminergic GPCR ligand design.
Hogendorf AS, Hogendorf A, Kurczab R, Kalinowska-Tłuścik J, Popik P, Nikiforuk A, Krawczyk M, Satała G, Lenda T, Knutelska J, Bugno R, Staroń J, Pietruś W, Matłoka M, Dubiel K, Moszczyński-Pętkowski R, Pieczykolan J, Wieczorek M, Pilarski B, Zajdel P, Bojarski AJ.
Hogendorf AS, et al. Among authors: moszczynski petkowski r.
Eur J Med Chem. 2019 Oct 1;179:1-15. doi: 10.1016/j.ejmech.2019.06.001. Epub 2019 Jun 5.
Eur J Med Chem. 2019.
PMID: 31229883
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