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Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications.
Nat Chem. 2021 Jun;13(6):540-548. doi: 10.1038/s41557-021-00660-y. Epub 2021 Apr 8.
Nat Chem. 2021.
PMID: 33833446
Free PMC article.
Publisher Correction: Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications.
Favalli N, Bassi G, Pellegrino C, Millul J, De Luca R, Cazzamalli S, Yang S, Trenner A, Mozaffari NL, Myburgh R, Moroglu M, Conway SJ, Sartori AA, Manz MG, Lerner RA, Vogt PK, Scheuermann J, Neri D.
Favalli N, et al. Among authors: moroglu m.
Nat Chem. 2021 Jul;13(7):714. doi: 10.1038/s41557-021-00742-x.
Nat Chem. 2021.
PMID: 34103693
No abstract available.
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Selective Fragments for the CREBBP Bromodomain Identified from an Encoded Self-assembly Chemical Library.
Catalano M, Moroglu M, Balbi P, Mazzieri F, Clayton J, Andrews KH, Bigatti M, Scheuermann J, Conway SJ, Neri D.
Catalano M, et al. Among authors: moroglu m.
ChemMedChem. 2020 Sep 16;15(18):1752-1756. doi: 10.1002/cmdc.202000528. Epub 2020 Aug 19.
ChemMedChem. 2020.
PMID: 32686307
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A Single-Stranded DNA-Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks.
Bassi G, Favalli N, Vuk M, Catalano M, Martinelli A, Trenner A, Porro A, Yang S, Tham CL, Moroglu M, Yue WW, Conway SJ, Vogt PK, Sartori AA, Scheuermann J, Neri D.
Bassi G, et al. Among authors: moroglu m.
Adv Sci (Weinh). 2020 Oct 14;7(22):2001970. doi: 10.1002/advs.202001970. eCollection 2020 Nov.
Adv Sci (Weinh). 2020.
PMID: 33240760
Free PMC article.
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Chemical Epigenetics: The Impact of Chemical and Chemical Biology Techniques on Bromodomain Target Validation.
Schiedel M, Moroglu M, Ascough DMH, Chamberlain AER, Kamps JJAG, Sekirnik AR, Conway SJ.
Schiedel M, et al. Among authors: moroglu m.
Angew Chem Int Ed Engl. 2019 Dec 9;58(50):17930-17952. doi: 10.1002/anie.201812164. Epub 2019 Nov 14.
Angew Chem Int Ed Engl. 2019.
PMID: 30633431
Review.
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Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain.
Brand M, Clayton J, Moroglu M, Schiedel M, Picaud S, Bluck JP, Skwarska A, Bolland H, Chan AKN, Laurin CMC, Scorah AR, See L, Rooney TPC, Andrews KH, Fedorov O, Perell G, Kalra P, Vinh KB, Cortopassi WA, Heitel P, Christensen KE, Cooper RI, Paton RS, Pomerantz WCK, Biggin PC, Hammond EM, Filippakopoulos P, Conway SJ.
Brand M, et al. Among authors: moroglu m.
J Med Chem. 2021 Jul 22;64(14):10102-10123. doi: 10.1021/acs.jmedchem.1c00348. Epub 2021 Jul 13.
J Med Chem. 2021.
PMID: 34255515
Free PMC article.
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BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability.
Jennings LE, Schiedel M, Hewings DS, Picaud S, Laurin CMC, Bruno PA, Bluck JP, Scorah AR, See L, Reynolds JK, Moroglu M, Mistry IN, Hicks A, Guzanov P, Clayton J, Evans CNG, Stazi G, Biggin PC, Mapp AK, Hammond EM, Humphreys PG, Filippakopoulos P, Conway SJ.
Jennings LE, et al. Among authors: moroglu m.
Bioorg Med Chem. 2018 Jul 15;26(11):2937-2957. doi: 10.1016/j.bmc.2018.05.003. Epub 2018 May 15.
Bioorg Med Chem. 2018.
PMID: 29776834
Free article.
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