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Aminoazabenzimidazoles, a novel class of orally active antimalarial agents.
J Med Chem. 2014 Jul 10;57(13):5702-13. doi: 10.1021/jm500535j. Epub 2014 Jun 24.
J Med Chem. 2014.
PMID: 24914738
Diarylthiazole: an antimycobacterial scaffold potentially targeting PrrB-PrrA two-component system.
Bellale E, Naik M, V B V, Ambady A, Narayan A, Ravishankar S, Ramachandran V, Kaur P, McLaughlin R, Whiteaker J, Morayya S, Guptha S, Sharma S, Raichurkar A, Awasthy D, Achar V, Vachaspati P, Bandodkar B, Panda M, Chatterji M.
Bellale E, et al. Among authors: morayya s.
J Med Chem. 2014 Aug 14;57(15):6572-82. doi: 10.1021/jm500833f. Epub 2014 Jul 16.
J Med Chem. 2014.
PMID: 24967731
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N-aryl-2-aminobenzimidazoles: novel, efficacious, antimalarial lead compounds.
Ramachandran S, Hameed P S, Srivastava A, Shanbhag G, Morayya S, Rautela N, Awasthy D, Kavanagh S, Bharath S, Reddy J, Panduga V, Prabhakar KR, Saralaya R, Nanduri R, Raichurkar A, Menasinakai S, Achar V, Jiménez-Díaz MB, Martínez MS, Angulo-Barturen I, Ferrer S, Sanz LM, Gamo FJ, Duffy S, Avery VM, Waterson D, Lee MC, Coburn-Flynn O, Fidock DA, Iyer PS, Narayanan S, Hosagrahara V, Sambandamurthy VK.
Ramachandran S, et al. Among authors: morayya s.
J Med Chem. 2014 Aug 14;57(15):6642-52. doi: 10.1021/jm500715u. Epub 2014 Jul 21.
J Med Chem. 2014.
PMID: 25007124
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Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate.
Hameed P S, Solapure S, Patil V, Henrich PP, Magistrado PA, Bharath S, Murugan K, Viswanath P, Puttur J, Srivastava A, Bellale E, Panduga V, Shanbag G, Awasthy D, Landge S, Morayya S, Koushik K, Saralaya R, Raichurkar A, Rautela N, Roy Choudhury N, Ambady A, Nandishaiah R, Reddy J, Prabhakar KR, Menasinakai S, Rudrapatna S, Chatterji M, Jiménez-Díaz MB, Martínez MS, Sanz LM, Coburn-Flynn O, Fidock DA, Lukens AK, Wirth DF, Bandodkar B, Mukherjee K, McLaughlin RE, Waterson D, Rosenbrier-Ribeiro L, Hickling K, Balasubramanian V, Warner P, Hosagrahara V, Dudley A, Iyer PS, Narayanan S, Kavanagh S, Sambandamurthy VK.
Hameed P S, et al. Among authors: morayya s.
Nat Commun. 2015 Mar 31;6:6715. doi: 10.1038/ncomms7715.
Nat Commun. 2015.
PMID: 25823686
Free PMC article.
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Development of a rapid and reliable assay for in vitro determination of compound cidality against the asexual stages of Plasmodium falciparum.
Viswanath P, Morayya S, Rautela N, Sinha A.
Viswanath P, et al. Among authors: morayya s.
Acta Parasitol. 2016 Dec 1;61(4):828-835. doi: 10.1515/ap-2016-0115.
Acta Parasitol. 2016.
PMID: 27787213
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Roles of the two type II NADH dehydrogenases in the survival of Mycobacterium tuberculosis in vitro.
Awasthy D, Ambady A, Narayana A, Morayya S, Sharma U.
Awasthy D, et al. Among authors: morayya s.
Gene. 2014 Oct 15;550(1):110-6. doi: 10.1016/j.gene.2014.08.024. Epub 2014 Aug 13.
Gene. 2014.
PMID: 25128581
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Revisiting the essentiality of glutamate racemase in Mycobacterium tuberculosis.
Morayya S, Awasthy D, Yadav R, Ambady A, Sharma U.
Morayya S, et al.
Gene. 2015 Jan 25;555(2):269-76. doi: 10.1016/j.gene.2014.11.017. Epub 2014 Nov 12.
Gene. 2015.
PMID: 25447907
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