Montgomery AP - Search Results

1

DYRK1A Negatively Regulates CDK5-SOX2 Pathway and Self-Renewal of Glioblastoma Stem Cells.

Chen B, McCuaig-Walton D, Tan S, Montgomery AP, Day BW, Kassiou M, Munoz L, Recasens A. Chen B, et al. Among authors: montgomery ap. Int J Mol Sci. 2021 Apr 13;22(8):4011. doi: 10.3390/ijms22084011. Int J Mol Sci. 2021. PMID: 33924599 Free PMC article.

2

Tricyclic heterocycles display diverse sensitivity to the A147T TSPO polymorphism.

Sokias R, Werry EL, Alison Cheng HW, Lloyd JH, Sohler G, Danon JJ, Montgomery AP, Du JJ, Gao Q, Hibbs DE, Ittner LM, Reekie TA, Kassiou M. Sokias R, et al. Among authors: montgomery ap. Eur J Med Chem. 2020 Dec 1;207:112725. doi: 10.1016/j.ejmech.2020.112725. Epub 2020 Aug 15. Eur J Med Chem. 2020. PMID: 32920427

3

The discovery of a potent and selective pyrazolo-[2,3-e]-[1,2,4]-triazine cannabinoid type 2 receptor agonist.

Moir M, Lane S, Montgomery AP, Hibbs D, Connor M, Kassiou M. Moir M, et al. Among authors: montgomery ap. Eur J Med Chem. 2021 Jan 15;210:113087. doi: 10.1016/j.ejmech.2020.113087. Epub 2020 Dec 5. Eur J Med Chem. 2021. PMID: 33321261

4

Strategies for targeting the P2Y₁₂ receptor in the central nervous system.

Ma BB, Montgomery AP, Chen B, Kassiou M, Danon JJ. Ma BB, et al. Among authors: montgomery ap. Bioorg Med Chem Lett. 2022 Sep 1;71:128837. doi: 10.1016/j.bmcl.2022.128837. Epub 2022 May 28. Bioorg Med Chem Lett. 2022. PMID: 35640763 Review.

5

Recent Scaffold Hopping Applications in Central Nervous System Drug Discovery.

Callis TB, Garrett TR, Montgomery AP, Danon JJ, Kassiou M. Callis TB, et al. Among authors: montgomery ap. J Med Chem. 2022 Oct 27;65(20):13483-13504. doi: 10.1021/acs.jmedchem.2c00969. Epub 2022 Oct 7. J Med Chem. 2022. PMID: 36206553 Review.

6

Understanding In Vitro Pathways to Drug Discovery for TDP-43 Proteinopathies.

Cheng HWA, Callis TB, Montgomery AP, Danon JJ, Jorgensen WT, Ke YD, Ittner LM, Werry EL, Kassiou M. Cheng HWA, et al. Among authors: montgomery ap. Int J Mol Sci. 2022 Nov 25;23(23):14769. doi: 10.3390/ijms232314769. Int J Mol Sci. 2022. PMID: 36499097 Free PMC article.

7

An update on late-stage functionalization in today's drug discovery.

Montgomery AP, Joyce JM, Danon JJ, Kassiou M. Montgomery AP, et al. Expert Opin Drug Discov. 2023 Jun;18(6):597-613. doi: 10.1080/17460441.2023.2205635. Epub 2023 Apr 28. Expert Opin Drug Discov. 2023. PMID: 37114995 Review.

8

Late-stage Functionalization for Improving Drug-like Molecular Properties.

Castellino NJ, Montgomery AP, Danon JJ, Kassiou M. Castellino NJ, et al. Among authors: montgomery ap. Chem Rev. 2023 Jul 12;123(13):8127-8153. doi: 10.1021/acs.chemrev.2c00797. Epub 2023 Jun 7. Chem Rev. 2023. PMID: 37285604 Review.

9

Synthesis and Preclinical Evaluation of Fluorinated 5-Azaindoles as CB2 PET Radioligands.

Kallinen A, Mardon K, Lane S, Montgomery AP, Bhalla R, Stimson DHR, Ahamed M, Cowin GJ, Hibbs D, Werry EL, Fulton R, Connor M, Kassiou M. Kallinen A, et al. Among authors: montgomery ap. ACS Chem Neurosci. 2023 Aug 16;14(16):2902-2921. doi: 10.1021/acschemneuro.3c00345. Epub 2023 Jul 27. ACS Chem Neurosci. 2023. PMID: 37499194

10

Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia.

Carey-Smith SL, Simad MH, Panchal K, Aya-Bonilla C, Smolders H, Lin S, Armitage JD, Nguyen VT, Bentley K, Ford J, Singh S, Oommen J, Laurent AP, Mercher T, Crispino JD, Montgomery AP, Kassiou M, Besson T, Deau E, Meijer L, Cheung LC, Kotecha RS, Malinge S. Carey-Smith SL, et al. Among authors: montgomery ap. Haematologica. 2024 Feb 29. doi: 10.3324/haematol.2023.284271. Online ahead of print. Haematologica. 2024. PMID: 38426275 Free article.

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