Mitsuya H - Search Results

1

Indole Chloropyridinyl Ester-Derived SARS-CoV-2 3CLpro Inhibitors: Enzyme Inhibition, Antiviral Efficacy, Structure-Activity Relationship, and X-ray Structural Studies.

Ghosh AK, Raghavaiah J, Shahabi D, Yadav M, Anson BJ, Lendy EK, Hattori SI, Higashi-Kuwata N, Mitsuya H, Mesecar AD. Ghosh AK, et al. Among authors: mitsuya h. J Med Chem. 2021 Oct 14;64(19):14702-14714. doi: 10.1021/acs.jmedchem.1c01214. Epub 2021 Sep 16. J Med Chem. 2021. PMID: 34528437 Free PMC article.

2

Chemistry and anti-HIV properties of 2'-fluoro-2',3'-dideoxyarabinofuranosylpyrimidines.

Siddiqui MA, Driscoll JS, Marquez VE, Roth JS, Shirasaka T, Mitsuya H, Barchi JJ Jr, Kelley JA. Siddiqui MA, et al. Among authors: mitsuya h. J Med Chem. 1992 Jun 12;35(12):2195-201. doi: 10.1021/jm00090a008. J Med Chem. 1992. PMID: 1351945

3

A ring-enlarged oxetanocin A analogue as an inhibitor of HIV infectivity.

Tseng CK, Marquez VE, Milne GW, Wysocki RJ Jr, Mitsuya H, Shirasaki T, Driscoll JS. Tseng CK, et al. Among authors: mitsuya h. J Med Chem. 1991 Jan;34(1):343-9. doi: 10.1021/jm00105a054. J Med Chem. 1991. PMID: 1992135

4

Potential anti-AIDS drugs. Lipophilic, adenosine deaminase-activated prodrugs.

Barchi JJ Jr, Marquez VE, Driscoll JS, Ford H Jr, Mitsuya H, Shirasaka T, Aoki S, Kelley JA. Barchi JJ Jr, et al. Among authors: mitsuya h. J Med Chem. 1991 May;34(5):1647-55. doi: 10.1021/jm00109a018. J Med Chem. 1991. PMID: 2033591

5

Conformationally locked nucleoside analogues. Synthesis of dideoxycarbocyclic nucleoside analogues structurally related to neplanocin C.

Rodriguez JB, Marquez VE, Nicklaus MC, Mitsuya H, Barchi JJ Jr. Rodriguez JB, et al. Among authors: mitsuya h. J Med Chem. 1994 Sep 30;37(20):3389-99. doi: 10.1021/jm00046a024. J Med Chem. 1994. PMID: 7932567

6

Lipophilic, acid-stable, adenosine deaminase-activated anti-HIV prodrugs for central nervous system delivery. 3. 6-Amino prodrugs of 2'-beta-fluoro-2',3'-dideoxyinosine.

Driscoll JS, Siddiqui MA, Ford H Jr, Kelley JA, Roth JS, Mitsuya H, Tanaka M, Marquez VE. Driscoll JS, et al. Among authors: mitsuya h. J Med Chem. 1996 Apr 12;39(8):1619-25. doi: 10.1021/jm9509197. J Med Chem. 1996. PMID: 8648601

7

A potent human immunodeficiency virus type 1 protease inhibitor, UIC-94003 (TMC-126), and selection of a novel (A28S) mutation in the protease active site.

Yoshimura K, Kato R, Kavlick MF, Nguyen A, Maroun V, Maeda K, Hussain KA, Ghosh AK, Gulnik SV, Erickson JW, Mitsuya H. Yoshimura K, et al. Among authors: mitsuya h. J Virol. 2002 Feb;76(3):1349-58. doi: 10.1128/jvi.76.3.1349-1358.2002. J Virol. 2002. PMID: 11773409 Free PMC article.

8

A conformationally locked analogue of the anti-HIV agent stavudine. An important correlation between pseudorotation and maximum amplitude.

Choi Y, George C, Comin MJ, Barchi JJ Jr, Kim HS, Jacobson KA, Balzarini J, Mitsuya H, Boyer PL, Hughes SH, Marquez VE. Choi Y, et al. Among authors: mitsuya h. J Med Chem. 2003 Jul 17;46(15):3292-9. doi: 10.1021/jm030116g. J Med Chem. 2003. PMID: 12852759

9

Novel bis-tetrahydrofuranylurethane-containing nonpeptidic protease inhibitor (PI) UIC-94017 (TMC114) with potent activity against multi-PI-resistant human immunodeficiency virus in vitro.

Koh Y, Nakata H, Maeda K, Ogata H, Bilcer G, Devasamudram T, Kincaid JF, Boross P, Wang YF, Tie Y, Volarath P, Gaddis L, Harrison RW, Weber IT, Ghosh AK, Mitsuya H. Koh Y, et al. Among authors: mitsuya h. Antimicrob Agents Chemother. 2003 Oct;47(10):3123-9. doi: 10.1128/AAC.47.10.3123-3129.2003. Antimicrob Agents Chemother. 2003. PMID: 14506019 Free PMC article.

10

A 4'-C-ethynyl-2',3'-dideoxynucleoside analogue highlights the role of the 3'-OH in anti-HIV active 4'-C-ethynyl-2'-deoxy nucleosides.

Siddiqui MA, Hughes SH, Boyer PL, Mitsuya H, Van QN, George C, Sarafinanos SG, Marquez VE. Siddiqui MA, et al. Among authors: mitsuya h. J Med Chem. 2004 Oct 7;47(21):5041-8. doi: 10.1021/jm049550o. J Med Chem. 2004. PMID: 15456247

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

710 results

Search Page