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Proximity-Induced Nucleic Acid Degrader (PINAD) Approach to Targeted RNA Degradation Using Small Molecules.
ACS Cent Sci. 2023 Apr 26;9(5):892-904. doi: 10.1021/acscentsci.3c00015. eCollection 2023 May 24.
ACS Cent Sci. 2023.
PMID: 37252343
Free PMC article.
meCLICK-Seq, a Substrate-Hijacking and RNA Degradation Strategy for the Study of RNA Methylation.
Mikutis S, Gu M, Sendinc E, Hazemi ME, Kiely-Collins H, Aspris D, Vassiliou GS, Shi Y, Tzelepis K, Bernardes GJL.
Mikutis S, et al.
ACS Cent Sci. 2020 Dec 23;6(12):2196-2208. doi: 10.1021/acscentsci.0c01094. Epub 2020 Oct 29.
ACS Cent Sci. 2020.
PMID: 33376781
Free PMC article.
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SnapShot: Clinical and preclinical utility of click chemistry.
Mikutis S, Bernardes GJL.
Mikutis S, et al.
Cell. 2023 Feb 2;186(3):662-662.e1. doi: 10.1016/j.cell.2023.01.018.
Cell. 2023.
PMID: 36736302
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METTL1-mediated m7G modification of Arg-TCT tRNA drives oncogenic transformation.
Orellana EA, Liu Q, Yankova E, Pirouz M, De Braekeleer E, Zhang W, Lim J, Aspris D, Sendinc E, Garyfallos DA, Gu M, Ali R, Gutierrez A, Mikutis S, Bernardes GJL, Fischer ES, Bradley A, Vassiliou GS, Slack FJ, Tzelepis K, Gregory RI.
Orellana EA, et al. Among authors: mikutis s.
Mol Cell. 2021 Aug 19;81(16):3323-3338.e14. doi: 10.1016/j.molcel.2021.06.031. Epub 2021 Aug 4.
Mol Cell. 2021.
PMID: 34352207
Free PMC article.
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Controlled masking and targeted release of redox-cycling ortho-quinones via a C-C bond-cleaving 1,6-elimination.
Dunsmore L, Navo CD, Becher J, de Montes EG, Guerreiro A, Hoyt E, Brown L, Zelenay V, Mikutis S, Cooper J, Barbieri I, Lawrinowitz S, Siouve E, Martin E, Ruivo PR, Rodrigues T, da Cruz FP, Werz O, Vassiliou G, Ravn P, Jiménez-Osés G, Bernardes GJL.
Dunsmore L, et al. Among authors: mikutis s.
Nat Chem. 2022 Jul;14(7):754-765. doi: 10.1038/s41557-022-00964-7. Epub 2022 Jun 27.
Nat Chem. 2022.
PMID: 35764792
Free PMC article.
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Orthogonal Stimuli Trigger Self-Assembly and Phase Transfer of FeII4L4 Cages and Cargoes.
McConnell AJ, Haynes CJE, Grommet AB, Aitchison CM, Guilleme J, Mikutis S, Nitschke JR.
McConnell AJ, et al. Among authors: mikutis s.
J Am Chem Soc. 2018 Dec 12;140(49):16952-16956. doi: 10.1021/jacs.8b11324. Epub 2018 Nov 30.
J Am Chem Soc. 2018.
PMID: 30465601
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Machine Learning Uncovers Natural Product Modulators of the 5-Lipoxygenase Pathway and Facilitates the Elucidation of Their Biological Mechanisms.
Mikutis S, Lawrinowitz S, Kretzer C, Dunsmore L, Sketeris L, Rodrigues T, Werz O, Bernardes GJL.
Mikutis S, et al.
ACS Chem Biol. 2024 Jan 19;19(1):217-229. doi: 10.1021/acschembio.3c00725. Epub 2023 Dec 27.
ACS Chem Biol. 2024.
PMID: 38149598
Free PMC article.
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