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Synthesis of Novel Benzenesulfonamide-Bearing Functionalized Imidazole Derivatives as Novel Candidates Targeting Multidrug-Resistant Mycobacterium abscessus Complex.
Balandis B, Kavaliauskas P, Grybaitė B, Petraitis V, Petraitienė R, Naing E, Garcia A, Grigalevičiūtė R, Mickevičius V. Balandis B, et al. Among authors: mickevicius v. Microorganisms. 2023 Apr 3;11(4):935. doi: 10.3390/microorganisms11040935. Microorganisms. 2023. PMID: 37110358 Free PMC article.
Synthesis, ADMET Properties, and In Vitro Antimicrobial and Antibiofilm Activity of 5-Nitro-2-thiophenecarbaldehyde N-((E)-(5-Nitrothienyl)methylidene)hydrazone (KTU-286) against Staphylococcus aureus with Defined Resistance Mechanisms.
Kavaliauskas P, Grybaite B, Mickevicius V, Petraitiene R, Grigaleviciute R, Planciuniene R, Gialanella P, Pockevicius A, Petraitis V. Kavaliauskas P, et al. Among authors: mickevicius v. Antibiotics (Basel). 2020 Sep 17;9(9):612. doi: 10.3390/antibiotics9090612. Antibiotics (Basel). 2020. PMID: 32957471 Free PMC article.
Synthesis of Novel Thiazole Derivatives Bearing β-Amino Acid and Aromatic Moieties as Promising Scaffolds for the Development of New Antibacterial and Antifungal Candidates Targeting Multidrug-Resistant Pathogens.
Malūkaitė D, Grybaitė B, Vaickelionienė R, Vaickelionis G, Sapijanskaitė-Banevič B, Kavaliauskas P, Mickevičius V. Malūkaitė D, et al. Among authors: mickevicius v. Molecules. 2021 Dec 23;27(1):74. doi: 10.3390/molecules27010074. Molecules. 2021. PMID: 35011308 Free PMC article.
Beta and Gamma Amino Acid-Substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases.
Balandis B, Šimkūnas T, Paketurytė-Latvė V, Michailovienė V, Mickevičiūtė A, Manakova E, Gražulis S, Belyakov S, Kairys V, Mickevičius V, Zubrienė A, Matulis D. Balandis B, et al. Among authors: mickevicius v. Pharmaceuticals (Basel). 2022 Apr 13;15(4):477. doi: 10.3390/ph15040477. Pharmaceuticals (Basel). 2022. PMID: 35455474 Free PMC article.
Synthesis, Biological Activity, and Molecular Modelling Studies of Naphthoquinone Derivatives as Promising Anticancer Candidates Targeting COX-2.
Kavaliauskas P, Opazo FS, Acevedo W, Petraitiene R, Grybaitė B, Anusevičius K, Mickevičius V, Belyakov S, Petraitis V. Kavaliauskas P, et al. Among authors: mickevicius v. Pharmaceuticals (Basel). 2022 Apr 27;15(5):541. doi: 10.3390/ph15050541. Pharmaceuticals (Basel). 2022. PMID: 35631366 Free PMC article.
28 results