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Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump.
Eur J Med Chem. 2023 Nov 5;259:115630. doi: 10.1016/j.ejmech.2023.115630. Epub 2023 Jul 7.
Eur J Med Chem. 2023.
PMID: 37459793
Free article.
Pyridylpiperazine efflux pump inhibitor boosts in vivo antibiotic efficacy against K. pneumoniae.
Vieira Da Cruz A, Jiménez-Castellanos JC, Börnsen C, Van Maele L, Compagne N, Pradel E, Müller RT, Meurillon V, Soulard D, Piveteau C, Biela A, Dumont J, Leroux F, Deprez B, Willand N, Pos KM, Frangakis AS, Hartkoorn RC, Flipo M.
Vieira Da Cruz A, et al. Among authors: meurillon v.
EMBO Mol Med. 2024 Jan;16(1):93-111. doi: 10.1038/s44321-023-00007-9. Epub 2023 Dec 20.
EMBO Mol Med. 2024.
PMID: 38177534
Free PMC article.
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