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Page 1
Identification of a sirtuin 3 inhibitor that displays selectivity over sirtuin 1 and 2.
Eur J Med Chem. 2012 Sep;55:58-66. doi: 10.1016/j.ejmech.2012.07.001. Epub 2012 Jul 15.
Eur J Med Chem. 2012.
PMID: 22835719
Replacement of the double bond of antitubulin chalcones with triazoles and tetrazoles: Synthesis and biological evaluation.
Mesenzani O, Massarotti A, Giustiniano M, Pirali T, Bevilacqua V, Caldarelli A, Canonico P, Sorba G, Novellino E, Genazzani AA, Tron GC.
Mesenzani O, et al.
Bioorg Med Chem Lett. 2011 Jan 15;21(2):764-8. doi: 10.1016/j.bmcl.2010.11.113. Epub 2010 Nov 28.
Bioorg Med Chem Lett. 2011.
PMID: 21167709
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Anthracycline-induced cardiotoxicity: A multicenter randomised trial comparing two strategies for guiding prevention with enalapril: The International CardioOncology Society-one trial.
Cardinale D, Ciceri F, Latini R, Franzosi MG, Sandri MT, Civelli M, Cucchi G, Menatti E, Mangiavacchi M, Cavina R, Barbieri E, Gori S, Colombo A, Curigliano G, Salvatici M, Rizzo A, Ghisoni F, Bianchi A, Falci C, Aquilina M, Rocca A, Monopoli A, Milandri C, Rossetti G, Bregni M, Sicuro M, Malossi A, Nassiacos D, Verusio C, Giordano M, Staszewsky L, Barlera S, Nicolis EB, Magnoli M, Masson S, Cipolla CM; ICOS-ONE Study Investigators.
Cardinale D, et al.
Eur J Cancer. 2018 May;94:126-137. doi: 10.1016/j.ejca.2018.02.005. Epub 2018 Mar 20.
Eur J Cancer. 2018.
PMID: 29567630
Clinical Trial.
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Identification of novel antitubulin agents by using a virtual screening approach based on a 7-point pharmacophore model of the tubulin colchi-site.
Massarotti A, Theeramunkong S, Mesenzani O, Caldarelli A, Genazzani AA, Tron GC.
Massarotti A, et al. Among authors: mesenzani o.
Chem Biol Drug Des. 2011 Dec;78(6):913-22. doi: 10.1111/j.1747-0285.2011.01245.x. Epub 2011 Oct 31.
Chem Biol Drug Des. 2011.
PMID: 22039890
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