Mesaros EF - Search Results

1

Design, synthesis, and binding affinities of pyrrolinone-based somatostatin mimetics.

Smith AB 3rd, Charnley AK, Mesaros EF, Kikuchi O, Wang W, Benowitz A, Chu CL, Feng JJ, Chen KH, Lin A, Cheng FC, Taylor L, Hirschmann R. Smith AB 3rd, et al. Among authors: mesaros ef. Org Lett. 2005 Feb 3;7(3):399-402. doi: 10.1021/ol0476974. Org Lett. 2005. PMID: 15673249

2

Design, synthesis, and structural analysis of D,L-mixed polypyrrolinones. 2. Macrocyclic hexapyrrolinones.

Smith AB 3rd, Xiong H, Charnley AK, Brenner M, Mesaros EF, Kenesky CS, Di Costanzo L, Christianson DW, Hirschmann R. Smith AB 3rd, et al. Among authors: mesaros ef. Org Lett. 2010 Jul 2;12(13):2994-7. doi: 10.1021/ol101008y. Org Lett. 2010. PMID: 20518572 Free PMC article.

3

Total synthesis of (-)-kendomycin exploiting a Petasis-Ferrier rearrangement/ring-closing olefin metathesis synthetic strategy.

Smith AB 3rd, Mesaros EF, Meyer EA. Smith AB 3rd, et al. Among authors: mesaros ef. J Am Chem Soc. 2005 May 18;127(19):6948-9. doi: 10.1021/ja051420x. J Am Chem Soc. 2005. PMID: 15884927

4

Evolution of a total synthesis of (-)-kendomycin exploiting a Petasis-Ferrier rearrangement/ring-closing olefin metathesis strategy.

Smith AB 3rd, Mesaros EF, Meyer EA. Smith AB 3rd, et al. Among authors: mesaros ef. J Am Chem Soc. 2006 Apr 19;128(15):5292-9. doi: 10.1021/ja060369+. J Am Chem Soc. 2006. PMID: 16608366

5

Diastereoselective conjugate additions to pi-allylmolybdenum complexes: a stereocontrolled route to 3,4,5-trisubstituted gamma-butyrolactones.

Pearson AJ, Mesaros EF. Pearson AJ, et al. Among authors: mesaros ef. Org Lett. 2002 Jun 13;4(12):2001-4. doi: 10.1021/ol020043f. Org Lett. 2002. PMID: 12049502

6

Stereocontrolled construction of tetrahydrofurans and gamma-butyrolactones using organomolybdenum chemistry.

Pearson AJ, Mesaros EF. Pearson AJ, et al. Among authors: mesaros ef. Org Lett. 2001 Aug 23;3(17):2665-8. doi: 10.1021/ol010121j. Org Lett. 2001. PMID: 11506604

7

Methanesulfonamido-cyclohexylamine derivatives of 2,4-diaminopyrimidine as potent ALK inhibitors.

Zificsak CA, Theroff JP, Aimone LD, Angeles TS, Albom MS, Cheng M, Mesaros EF, Ott GR, Quail MR, Underiner TL, Wan W, Dorsey BD. Zificsak CA, et al. Among authors: mesaros ef. Bioorg Med Chem Lett. 2011 Jul 1;21(13):3877-80. doi: 10.1016/j.bmcl.2011.05.040. Epub 2011 May 18. Bioorg Med Chem Lett. 2011. PMID: 21632243

8

Piperidine-3,4-diol and piperidine-3-ol derivatives of pyrrolo[2,1-f][1,2,4]triazine as inhibitors of anaplastic lymphoma kinase.

Mesaros EF, Angeles TS, Albom MS, Wagner JC, Aimone LD, Wan W, Lu L, Huang Z, Olsen M, Kordwitz E, Haltiwanger RC, Landis AJ, Cheng M, Ruggeri BA, Ator MA, Dorsey BD, Ott GR. Mesaros EF, et al. Bioorg Med Chem Lett. 2015 Mar 1;25(5):1047-52. doi: 10.1016/j.bmcl.2015.01.019. Epub 2015 Jan 17. Bioorg Med Chem Lett. 2015. PMID: 25655723

9

2,7-disubstituted-pyrrolo[2,1-f][1,2,4]triazines: new variant of an old template and application to the discovery of anaplastic lymphoma kinase (ALK) inhibitors with in vivo antitumor activity.

Ott GR, Wells GJ, Thieu TV, Quail MR, Lisko JG, Mesaros EF, Gingrich DE, Ghose AK, Wan W, Lu L, Cheng M, Albom MS, Angeles TS, Huang Z, Aimone LD, Ator MA, Ruggeri BA, Dorsey BD. Ott GR, et al. Among authors: mesaros ef. J Med Chem. 2011 Sep 22;54(18):6328-41. doi: 10.1021/jm200758k. Epub 2011 Aug 22. J Med Chem. 2011. PMID: 21859094

10

Strategies to mitigate the bioactivation of 2-anilino-7-aryl-pyrrolo[2,1-f][1,2,4]triazines: identification of orally bioavailable, efficacious ALK inhibitors.

Mesaros EF, Thieu TV, Wells GJ, Zificsak CA, Wagner JC, Breslin HJ, Tripathy R, Diebold JL, McHugh RJ, Wohler AT, Quail MR, Wan W, Lu L, Huang Z, Albom MS, Angeles TS, Wells-Knecht KJ, Aimone LD, Cheng M, Ator MA, Ott GR, Dorsey BD. Mesaros EF, et al. J Med Chem. 2012 Jan 12;55(1):115-25. doi: 10.1021/jm2010767. Epub 2011 Dec 29. J Med Chem. 2012. PMID: 22141319

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