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Antileishmanial activity of 2-amino-thiophene derivative SB-200.
Sousa JPA, Sousa JMS, Rodrigues RRL, Nunes TAL, Machado YAA, Araujo AC, da Silva IGM, Barros-Cordeiro KB, Báo SN, Alves MMM, Mendonça-Junior FJB, Rodrigues KADF. Sousa JPA, et al. Among authors: mendonca junior fjb. Int Immunopharmacol. 2023 Oct;123:110750. doi: 10.1016/j.intimp.2023.110750. Epub 2023 Aug 1. Int Immunopharmacol. 2023. PMID: 37536181
2-Amino-thiophene derivatives present antileishmanial activity mediated by apoptosis and immunomodulation in vitro.
Rodrigues KA, Dias CN, Néris PL, Rocha Jda C, Scotti MT, Scotti L, Mascarenhas SR, Veras RC, de Medeiros IA, Keesen Tde S, de Oliveira TB, de Lima Mdo C, Balliano TL, de Aquino TM, de Moura RO, Mendonça Junior FJ, de Oliveira MR. Rodrigues KA, et al. Eur J Med Chem. 2015 Dec 1;106:1-14. doi: 10.1016/j.ejmech.2015.10.011. Epub 2015 Oct 17. Eur J Med Chem. 2015. PMID: 26513640
New thiophene-acridine compounds: Synthesis, antileishmanial activity, DNA binding, chemometric, and molecular docking studies.
de Lima Serafim V, Félix MB, Frade Silva DK, Rodrigues KADF, Andrade PN, de Almeida SMV, de Albuquerque Dos Santos S, de Oliveira JF, de Lima MDCA, Mendonça-Junior FJB, Scotti MT, de Oliveira MR, de Moura RO. de Lima Serafim V, et al. Chem Biol Drug Des. 2018 Jun;91(6):1141-1155. doi: 10.1111/cbdd.13176. Epub 2018 Mar 25. Chem Biol Drug Des. 2018. PMID: 29415325
Design, synthesis and pharmacological evaluation of CVIB, a codrug of carvacrol and ibuprofen as a novel anti-inflammatory agent.
de Oliveira Pedrosa Rolim M, de Almeida AR, da Rocha Pitta MG, de Melo Rêgo MJB, Quintans-Júnior LJ, de Souza Siqueira Quintans J, Heimfarth L, Scotti L, Scotti MT, da Cruz RMD, de Almeida RN, da Silva TG, de Oliveira JA, de Campos ML, Marchand P, Mendonça-Junior FJB. de Oliveira Pedrosa Rolim M, et al. Int Immunopharmacol. 2019 Nov;76:105856. doi: 10.1016/j.intimp.2019.105856. Epub 2019 Aug 31. Int Immunopharmacol. 2019. PMID: 31480005
Thiophene-Based Compounds with Potential Anti-Inflammatory Activity.
da Cruz RMD, Mendonça-Junior FJB, de Mélo NB, Scotti L, de Araújo RSA, de Almeida RN, de Moura RO. da Cruz RMD, et al. Pharmaceuticals (Basel). 2021 Jul 19;14(7):692. doi: 10.3390/ph14070692. Pharmaceuticals (Basel). 2021. PMID: 34358118 Free PMC article. Review.
Selene-Ethylenelacticamides and N-Aryl-Propanamides as Broad-Spectrum Leishmanicidal Agents.
de Sousa NF, da Silva Souza HD, de Menezes RPB, da Silva Alves F, Acevedo CAH, de Lima Nunes TA, Sessions ZL, Scotti L, Muratov EN, Mendonça-Junior FJB, da Franca Rodrigues KA, de Athayde Filho PF, Scotti MT. de Sousa NF, et al. Among authors: mendonca junior fjb. Pathogens. 2023 Jan 13;12(1):136. doi: 10.3390/pathogens12010136. Pathogens. 2023. PMID: 36678484 Free PMC article.
67 results