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New thiophene-acridine compounds: Synthesis, antileishmanial activity, DNA binding, chemometric, and molecular docking studies.
de Lima Serafim V, Félix MB, Frade Silva DK, Rodrigues KADF, Andrade PN, de Almeida SMV, de Albuquerque Dos Santos S, de Oliveira JF, de Lima MDCA, Mendonça-Junior FJB, Scotti MT, de Oliveira MR, de Moura RO. de Lima Serafim V, et al. Chem Biol Drug Des. 2018 Jun;91(6):1141-1155. doi: 10.1111/cbdd.13176. Epub 2018 Mar 25. Chem Biol Drug Des. 2018. PMID: 29415325
2-Amino-thiophene derivatives present antileishmanial activity mediated by apoptosis and immunomodulation in vitro.
Rodrigues KA, Dias CN, Néris PL, Rocha Jda C, Scotti MT, Scotti L, Mascarenhas SR, Veras RC, de Medeiros IA, Keesen Tde S, de Oliveira TB, de Lima Mdo C, Balliano TL, de Aquino TM, de Moura RO, Mendonça Junior FJ, de Oliveira MR. Rodrigues KA, et al. Eur J Med Chem. 2015 Dec 1;106:1-14. doi: 10.1016/j.ejmech.2015.10.011. Epub 2015 Oct 17. Eur J Med Chem. 2015. PMID: 26513640
Modulation of Drug Resistance in Staphylococcus aureus with Coumarin Derivatives.
de Araújo RS, Barbosa-Filho JM, Scotti MT, Scotti L, da Cruz RM, Falcão-Silva Vdos S, de Siqueira-Júnior JP, Mendonça-Junior FJ. de Araújo RS, et al. Scientifica (Cairo). 2016;2016:6894758. doi: 10.1155/2016/6894758. Epub 2016 Apr 19. Scientifica (Cairo). 2016. PMID: 27200211 Free PMC article.
Anticancer properties of thiophene derivatives in breast cancer MCF-7 cells.
Dos Santos FA, Pereira MC, de Oliveira TB, Mendonça Junior FJB, de Lima MDCA, Pitta MGDR, Pitta IDR, de Melo Rêgo MJB, da Rocha Pitta MG. Dos Santos FA, et al. Anticancer Drugs. 2018 Feb;29(2):157-166. doi: 10.1097/CAD.0000000000000581. Anticancer Drugs. 2018. PMID: 29256900
67 results