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Highly Selective Phosphatidylinositol 4-Kinase IIIβ Inhibitors and Structural Insight into Their Mode of Action.
J Med Chem. 2015 May 14;58(9):3767-93. doi: 10.1021/acs.jmedchem.5b00499. Epub 2015 May 4.
J Med Chem. 2015.
PMID: 25897704
Purine analogs as phosphatidylinositol 4-kinase IIIβ inhibitors.
Šála M, Kögler M, Plačková P, Mejdrová I, Hřebabecký H, Procházková E, Strunin D, Lee G, Birkus G, Weber J, Mertlíková-Kaiserová H, Nencka R.
Šála M, et al. Among authors: mejdrova i.
Bioorg Med Chem Lett. 2016 Jun 1;26(11):2706-12. doi: 10.1016/j.bmcl.2016.04.002. Epub 2016 Apr 5.
Bioorg Med Chem Lett. 2016.
PMID: 27090557
Free PMC article.
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Rational Design of Novel Highly Potent and Selective Phosphatidylinositol 4-Kinase IIIβ (PI4KB) Inhibitors as Broad-Spectrum Antiviral Agents and Tools for Chemical Biology.
Mejdrová I, Chalupská D, Plačková P, Müller C, Šála M, Klíma M, Baumlová A, Hřebabecký H, Procházková E, Dejmek M, Strunin D, Weber J, Lee G, Matoušová M, Mertlíková-Kaiserová H, Ziebuhr J, Birkus G, Boura E, Nencka R.
Mejdrová I, et al.
J Med Chem. 2017 Jan 12;60(1):100-118. doi: 10.1021/acs.jmedchem.6b01465. Epub 2016 Dec 22.
J Med Chem. 2017.
PMID: 28004945
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Fluorescent Inhibitors as Tools To Characterize Enzymes: Case Study of the Lipid Kinase Phosphatidylinositol 4-Kinase IIIβ (PI4KB).
Humpolickova J, Mejdrová I, Matousova M, Nencka R, Boura E.
Humpolickova J, et al. Among authors: mejdrova i.
J Med Chem. 2017 Jan 12;60(1):119-127. doi: 10.1021/acs.jmedchem.6b01466. Epub 2016 Dec 22.
J Med Chem. 2017.
PMID: 28004946
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A large scale high-throughput screen identifies chemical inhibitors of phosphatidylinositol 4-kinase type II alpha.
Sengupta N, Jović M, Barnaeva E, Kim DW, Hu X, Southall N, Dejmek M, Mejdrova I, Nencka R, Baumlova A, Chalupska D, Boura E, Ferrer M, Marugan J, Balla T.
Sengupta N, et al. Among authors: mejdrova i.
J Lipid Res. 2019 Mar;60(3):683-693. doi: 10.1194/jlr.D090159. Epub 2019 Jan 9.
J Lipid Res. 2019.
PMID: 30626625
Free PMC article.
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Discovery of the Hedgehog Pathway Inhibitor Pipinib that Targets PI4KIIIß.
Kremer L, Hennes E, Brause A, Ursu A, Robke L, Matsubayashi HT, Nihongaki Y, Flegel J, Mejdrová I, Eickhoff J, Baumann M, Nencka R, Janning P, Kordes S, Schöler HR, Sterneckert J, Inoue T, Ziegler S, Waldmann H.
Kremer L, et al. Among authors: mejdrova i.
Angew Chem Int Ed Engl. 2019 Nov 11;58(46):16617-16628. doi: 10.1002/anie.201907632. Epub 2019 Oct 4.
Angew Chem Int Ed Engl. 2019.
PMID: 31454140
Free PMC article.
Review.
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RNA-Templated Peptide Bond Formation Promotes L-Homochirality.
Węgrzyn E, Mejdrová I, Müller FM, Nainytė M, Escobar L, Carell T.
Węgrzyn E, et al. Among authors: mejdrova i.
Angew Chem Int Ed Engl. 2024 May 6;63(19):e202319235. doi: 10.1002/anie.202319235. Epub 2024 Apr 5.
Angew Chem Int Ed Engl. 2024.
PMID: 38407532
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Discovery of Novel Human Constitutive Androstane Receptor Agonists with the Imidazo[1,2-a]pyridine Structure.
Mejdrová I, Dušek J, Škach K, Stefela A, Skoda J, Chalupský K, Dohnalová K, Pavkova I, Kronenberger T, Rashidian A, Smutná L, Duchoslav V, Smutny T, Pávek P, Nencka R.
Mejdrová I, et al.
J Med Chem. 2023 Feb 23;66(4):2422-2456. doi: 10.1021/acs.jmedchem.2c01140. Epub 2023 Feb 9.
J Med Chem. 2023.
PMID: 36756805
Free PMC article.
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