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Optimization of Ligands Using Focused DNA-Encoded Libraries To Develop a Selective, Cell-Permeable CBX8 Chromodomain Inhibitor.
ACS Chem Biol. 2020 Jan 17;15(1):112-131. doi: 10.1021/acschembio.9b00654. Epub 2019 Dec 12.
ACS Chem Biol. 2020.
PMID: 31755685
Free PMC article.
Accelerated Structural Prediction of Flexible Protein-Ligand Complexes: The SLICE Method.
McFarlane JMB, Krause KD, Paci I.
McFarlane JMB, et al.
J Chem Inf Model. 2019 Dec 23;59(12):5263-5275. doi: 10.1021/acs.jcim.9b00688. Epub 2019 Nov 21.
J Chem Inf Model. 2019.
PMID: 31693362
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Selective Inhibition of CBX6: A Methyllysine Reader Protein in the Polycomb Family.
Milosevich N, Gignac MC, McFarlane J, Simhadri C, Horvath S, Daze KD, Croft CS, Dheri A, Quon TT, Douglas SF, Wulff JE, Paci I, Hof F.
Milosevich N, et al.
ACS Med Chem Lett. 2015 Dec 7;7(2):139-44. doi: 10.1021/acsmedchemlett.5b00378. eCollection 2016 Feb 11.
ACS Med Chem Lett. 2015.
PMID: 26985288
Free PMC article.
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Pan-specific and partially selective dye-labeled peptidic inhibitors of the polycomb paralog proteins.
Milosevich N, McFarlane J, Gignac MC, Li J, Brown TM, Wilson CR, Devorkin L, Croft CS, Hof R, Paci I, Lum JJ, Hof F.
Milosevich N, et al.
Bioorg Med Chem. 2020 Jan 1;28(1):115176. doi: 10.1016/j.bmc.2019.115176. Epub 2019 Nov 9.
Bioorg Med Chem. 2020.
PMID: 31753799
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Structural study of a small molecule receptor bound to dimethyllysine in lysozyme.
McGovern RE, Snarr BD, Lyons JA, McFarlane J, Whiting AL, Paci I, Hof F, Crowley PB.
McGovern RE, et al.
Chem Sci. 2015 Jan 1;6(1):442-449. doi: 10.1039/C4SC02383H.
Chem Sci. 2015.
PMID: 25530835
Free PMC article.
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THE STAGES OF THE PEPTIC HYDROLYSIS OF EGG ALBUMIN.
McFarlane J, Dunbar VE, Borsook H, Wasteneys H.
McFarlane J, et al.
J Gen Physiol. 1927 Jan 20;10(3):437-50. doi: 10.1085/jgp.10.3.437.
J Gen Physiol. 1927.
PMID: 19872335
Free PMC article.
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