Mazitschek R - Search Results

1

Synthesis and biological evaluation of Santacruzamate-A based analogues.

Randino R, Gazzerro P, Mazitschek R, Rodriquez M. Randino R, et al. Among authors: mazitschek r. Bioorg Med Chem. 2017 Dec 15;25(24):6486-6491. doi: 10.1016/j.bmc.2017.10.026. Epub 2017 Oct 20. Bioorg Med Chem. 2017. PMID: 29100734

2

Discovery of novel class of histone deacetylase inhibitors as potential anticancer agents.

El-Awady R, Saleh E, Hamoudi R, Ramadan WS, Mazitschek R, Nael MA, Elokely KM, Abou-Gharbia M, Childers WE, Srinivasulu V, Aloum L, Menon V, Al-Tel TH. El-Awady R, et al. Among authors: mazitschek r. Bioorg Med Chem. 2021 Jul 15;42:116251. doi: 10.1016/j.bmc.2021.116251. Epub 2021 Jun 8. Bioorg Med Chem. 2021. PMID: 34116381

3

In vivo PET imaging of histone deacetylases by 18F-suberoylanilide hydroxamic acid (18F-SAHA).

Hendricks JA, Keliher EJ, Marinelli B, Reiner T, Weissleder R, Mazitschek R. Hendricks JA, et al. Among authors: mazitschek r. J Med Chem. 2011 Aug 11;54(15):5576-82. doi: 10.1021/jm200620f. Epub 2011 Jul 18. J Med Chem. 2011. PMID: 21721525 Free PMC article.

4

Dissecting structure-activity-relationships of crebinostat: Brain penetrant HDAC inhibitors for neuroepigenetic regulation.

Ghosh B, Zhao WN, Reis SA, Patnaik D, Fass DM, Tsai LH, Mazitschek R, Haggarty SJ. Ghosh B, et al. Among authors: mazitschek r. Bioorg Med Chem Lett. 2016 Feb 15;26(4):1265-1271. doi: 10.1016/j.bmcl.2016.01.022. Epub 2016 Jan 11. Bioorg Med Chem Lett. 2016. PMID: 26804233 Free PMC article.

5

Identification and characterization of small molecule inhibitors of a class I histone deacetylase from Plasmodium falciparum.

Patel V, Mazitschek R, Coleman B, Nguyen C, Urgaonkar S, Cortese J, Barker RH, Greenberg E, Tang W, Bradner JE, Schreiber SL, Duraisingh MT, Wirth DF, Clardy J. Patel V, et al. Among authors: mazitschek r. J Med Chem. 2009 Apr 23;52(8):2185-7. doi: 10.1021/jm801654y. J Med Chem. 2009. PMID: 19317450 Free PMC article.

6

Development of a fluorescence polarization based assay for histone deacetylase ligand discovery.

Mazitschek R, Patel V, Wirth DF, Clardy J. Mazitschek R, et al. Bioorg Med Chem Lett. 2008 May 1;18(9):2809-12. doi: 10.1016/j.bmcl.2008.04.007. Epub 2008 Apr 7. Bioorg Med Chem Lett. 2008. PMID: 18430569 Free PMC article.

7

Synthesis and antiplasmodial activity of novel 2,4-diaminopyrimidines.

Martyn DC, Nijjar A, Celatka CA, Mazitschek R, Cortese JF, Tyndall E, Liu H, Fitzgerald MM, O'Shea TJ, Danthi S, Clardy J. Martyn DC, et al. Among authors: mazitschek r. Bioorg Med Chem Lett. 2010 Jan 1;20(1):228-31. doi: 10.1016/j.bmcl.2009.10.133. Epub 2009 Oct 31. Bioorg Med Chem Lett. 2010. PMID: 19914064

8

Antiplasmodial activity of piperazine sulfonamides.

Martyn DC, Cortese JF, Tyndall E, Dick J, Mazitschek R, Munoz B, Clardy J. Martyn DC, et al. Among authors: mazitschek r. Bioorg Med Chem Lett. 2010 Jan 1;20(1):218-21. doi: 10.1016/j.bmcl.2009.10.130. Epub 2009 Oct 31. Bioorg Med Chem Lett. 2010. PMID: 19914069

9

Exploring the 3-piperidin-4-yl-1H-indole scaffold as a novel antimalarial chemotype.

Santos SA, Lukens AK, Coelho L, Nogueira F, Wirth DF, Mazitschek R, Moreira R, Paulo A. Santos SA, et al. Among authors: mazitschek r. Eur J Med Chem. 2015 Sep 18;102:320-33. doi: 10.1016/j.ejmech.2015.07.047. Epub 2015 Jul 31. Eur J Med Chem. 2015. PMID: 26295174

10

Selective HDAC inhibition by ACY-241 enhances the activity of paclitaxel in solid tumor models.

Huang P, Almeciga-Pinto I, Jarpe M, van Duzer JH, Mazitschek R, Yang M, Jones SS, Quayle SN. Huang P, et al. Among authors: mazitschek r. Oncotarget. 2017 Jan 10;8(2):2694-2707. doi: 10.18632/oncotarget.13738. Oncotarget. 2017. PMID: 27926524 Free PMC article.

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