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Synthesis, Kinetic and Conformational Studies of 2-Substituted-5-(β-d-glucopyranosyl)-pyrimidin-4-ones as Potential Inhibitors of Glycogen Phosphorylase.
Molecules. 2020 Nov 22;25(22):5463. doi: 10.3390/molecules25225463.
Molecules. 2020.
PMID: 33266408
Free PMC article.
A glucose-based molecular rotor inhibitor of glycogen phosphorylase as a probe of cellular enzymatic function.
Minadakis MP, Mavreas KF, Neofytos DD, Paschou M, Kogkaki A, Athanasiou V, Mamais M, Veclani D, Iatrou H, Venturini A, Chrysina ED, Papazafiri P, Gimisis T.
Minadakis MP, et al. Among authors: mavreas kf.
Org Biomol Chem. 2022 Mar 23;20(12):2407-2423. doi: 10.1039/d1ob02211c.
Org Biomol Chem. 2022.
PMID: 35119451
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Multiscale time-resolved fluorescence study of a glycogen phosphorylase inhibitor combined with quantum chemistry calculations.
Maffeis V , Mavreas K , Monti F , Mamais M , Gustavsson T , Chrysina ED , Markovitsi D , Gimisis T , Venturini A .
Maffeis V , et al.
Phys Chem Chem Phys. 2019 Apr 3;21(14):7685-7696. doi: 10.1039/c8cp07538g.
Phys Chem Chem Phys. 2019.
PMID: 30912774
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