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Identification of Inhibitors to Trypanosoma cruzi Sirtuins Based on Compounds Developed to Human Enzymes.
Int J Mol Sci. 2020 May 22;21(10):3659. doi: 10.3390/ijms21103659.
Int J Mol Sci. 2020.
PMID: 32455951
Free PMC article.
Sirtuin modulators: past, present, and future perspectives.
Fiorentino F, Mautone N, Menna M, D'Acunzo F, Mai A, Rotili D.
Fiorentino F, et al. Among authors: mautone n.
Future Med Chem. 2022 Jun;14(12):915-939. doi: 10.4155/fmc-2022-0031. Epub 2022 May 18.
Future Med Chem. 2022.
PMID: 35583203
Free PMC article.
Review.
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Sirtuin modulators: where are we now? A review of patents from 2015 to 2019.
Mautone N, Zwergel C, Mai A, Rotili D.
Mautone N, et al.
Expert Opin Ther Pat. 2020 Jun;30(6):389-407. doi: 10.1080/13543776.2020.1749264. Epub 2020 Apr 13.
Expert Opin Ther Pat. 2020.
PMID: 32228181
Review.
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Targeting histone acetylation/deacetylation in parasites: an update (2017-2020).
Fioravanti R, Mautone N, Rovere A, Rotili D, Mai A.
Fioravanti R, et al. Among authors: mautone n.
Curr Opin Chem Biol. 2020 Aug;57:65-74. doi: 10.1016/j.cbpa.2020.05.008. Epub 2020 Jun 29.
Curr Opin Chem Biol. 2020.
PMID: 32615359
Review.
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Recent advances in epigenetic proteolysis targeting chimeras (Epi-PROTACs).
Tomaselli D, Mautone N, Mai A, Rotili D.
Tomaselli D, et al. Among authors: mautone n.
Eur J Med Chem. 2020 Dec 1;207:112750. doi: 10.1016/j.ejmech.2020.112750. Epub 2020 Aug 18.
Eur J Med Chem. 2020.
PMID: 32871345
Review.
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First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.
Nowak RP, Tumber A, Hendrix E, Ansari MSZ, Sabatino M, Antonini L, Andrijes R, Salah E, Mautone N, Pellegrini FR, Simelis K, Kawamura A, Johansson C, Passeri D, Pellicciari R, Ciogli A, Del Bufalo D, Ragno R, Coleman ML, Trisciuoglio D, Mai A, Oppermann U, Schofield CJ, Rotili D.
Nowak RP, et al. Among authors: mautone n.
J Med Chem. 2021 Dec 9;64(23):17031-17050. doi: 10.1021/acs.jmedchem.1c00605. Epub 2021 Nov 29.
J Med Chem. 2021.
PMID: 34843649
Free PMC article.
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Tranylcypromine-Based LSD1 Inhibitors: Structure-Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation.
Fioravanti R, Romanelli A, Mautone N, Di Bello E, Rovere A, Corinti D, Zwergel C, Valente S, Rotili D, Botrugno OA, Dessanti P, Vultaggio S, Vianello P, Cappa A, Binda C, Mattevi A, Minucci S, Mercurio C, Varasi M, Mai A.
Fioravanti R, et al. Among authors: mautone n.
ChemMedChem. 2020 Apr 3;15(7):643-658. doi: 10.1002/cmdc.201900730. Epub 2020 Feb 14.
ChemMedChem. 2020.
PMID: 32003940
Free PMC article.
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From PARP1 to TNKS2 Inhibition: A Structure-Based Approach.
Tomassi S, Pfahler J, Mautone N, Rovere A, Esposito C, Passeri D, Pellicciari R, Novellino E, Pannek M, Steegborn C, Paiardini A, Mai A, Rotili D.
Tomassi S, et al. Among authors: mautone n.
ACS Med Chem Lett. 2020 Feb 3;11(5):862-868. doi: 10.1021/acsmedchemlett.9b00654. eCollection 2020 May 14.
ACS Med Chem Lett. 2020.
PMID: 32435397
Free PMC article.
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