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In vitro cytotoxicity and docking study of novel symmetric and asymmetric dihydropyridines and pyridines as EGFR tyrosine kinase inhibitors.
Chem Biol Drug Des. 2022 Jul;100(1):121-135. doi: 10.1111/cbdd.14058. Epub 2022 May 2.
Chem Biol Drug Des. 2022.
PMID: 35501997
Design, synthesis, and docking study of new quinoline derivatives as antitumor agents.
Nasr EE, Mostafa AS, El-Sayed MAA, Massoud MAM.
Nasr EE, et al. Among authors: massoud mam.
Arch Pharm (Weinheim). 2019 Jul;352(7):e1800355. doi: 10.1002/ardp.201800355. Epub 2019 May 13.
Arch Pharm (Weinheim). 2019.
PMID: 31081954
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Biological evaluation of newly synthesized quinoline-based compound PPQ-8 in acute and chronic toxoplasmosis: An experimental study.
Elgawad HA, Alhusseiny SM, Taman A, Youssef MY, Mansour B, Massoud M, Handousa A.
Elgawad HA, et al.
Exp Parasitol. 2019 Nov;206:107756. doi: 10.1016/j.exppara.2019.107756. Epub 2019 Sep 5.
Exp Parasitol. 2019.
PMID: 31494217
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Effect of a newly synthesized quinoline-based compound (PPQ-8) on murine schistosomiasis mansoni.
Taman A, Alhusseiny SM, Saleh NE, Youssef MY, Mansour B, Massoud M, El-Beshbishi SN.
Taman A, et al.
J Helminthol. 2020 Feb 7;94:e123. doi: 10.1017/S0022149X2000005X.
J Helminthol. 2020.
PMID: 32029011
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In vivo studies of the effect of PPQ-6, a quinoline-based agent against Schistosoma mansoni in mice.
Taman A, Alhusseiny SM, El-Zayady WM, Elblihy AA, Mansour B, Massoud M, Youssef MY, Saleh NE.
Taman A, et al.
Exp Parasitol. 2020 Aug;215:107933. doi: 10.1016/j.exppara.2020.107933. Epub 2020 Jun 7.
Exp Parasitol. 2020.
PMID: 32525006
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Benzimidazole-based protein kinase inhibitors: Current perspectives in targeted cancer therapy.
Ali AM, Tawfik SS, Mostafa AS, Massoud MAM.
Ali AM, et al. Among authors: massoud mam.
Chem Biol Drug Des. 2022 Nov;100(5):656-673. doi: 10.1111/cbdd.14130. Epub 2022 Aug 19.
Chem Biol Drug Des. 2022.
PMID: 35962624
Review.
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Modified Tacrine Derivatives as Multitarget-Directed Ligands for the Treatment of Alzheimer's Disease: Synthesis, Biological Evaluation, and Molecular Modeling Study.
Fares S, El Husseiny WM, Selim KB, Massoud MAM.
Fares S, et al. Among authors: massoud mam.
ACS Omega. 2023 Jul 12;8(29):26012-26034. doi: 10.1021/acsomega.3c02051. eCollection 2023 Jul 25.
ACS Omega. 2023.
PMID: 37521639
Free PMC article.
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