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Design, synthesis and stepwise optimization of nitrile-based inhibitors of cathepsins B and L.
Bioorg Med Chem. 2021 Jan 1;29:115827. doi: 10.1016/j.bmc.2020.115827. Epub 2020 Nov 16.
Bioorg Med Chem. 2021.
PMID: 33254069
Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor.
Ribeiro JFR, Cianni L, Li C, Warwick TG, de Vita D, Rosini F, Dos Reis Rocho F, Martins FCP, Kenny PW, Lameira J, Leitão A, Emsley J, Montanari CA.
Ribeiro JFR, et al. Among authors: martins fcp.
Bioorg Med Chem. 2020 Nov 15;28(22):115743. doi: 10.1016/j.bmc.2020.115743. Epub 2020 Sep 6.
Bioorg Med Chem. 2020.
PMID: 33038787
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