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Page 1
Adenosine receptors: what we know and what we are learning.
Trincavelli ML, Daniele S, Martini C. Trincavelli ML, et al. Among authors: martini c. Curr Top Med Chem. 2010;10(9):860-77. doi: 10.2174/156802610791268756. Curr Top Med Chem. 2010. PMID: 20370662 Review.
Frontal affinity chromatography-mass spectrometry useful for characterization of new ligands for GPR17 receptor.
Calleri E, Ceruti S, Cristalli G, Martini C, Temporini C, Parravicini C, Volpini R, Daniele S, Caccialanza G, Lecca D, Lambertucci C, Trincavelli ML, Marucci G, Wainer IW, Ranghino G, Fantucci P, Abbracchio MP, Massolini G. Calleri E, et al. Among authors: martini c. J Med Chem. 2010 May 13;53(9):3489-501. doi: 10.1021/jm901691y. J Med Chem. 2010. PMID: 20394377 Free PMC article.
Novel N2-substituted pyrazolo[3,4-d]pyrimidine adenosine A3 receptor antagonists: inhibition of A3-mediated human glioblastoma cell proliferation.
Taliani S, La Motta C, Mugnaini L, Simorini F, Salerno S, Marini AM, Da Settimo F, Cosconati S, Cosimelli B, Greco G, Limongelli V, Marinelli L, Novellino E, Ciampi O, Daniele S, Trincavelli ML, Martini C. Taliani S, et al. Among authors: martini c. J Med Chem. 2010 May 27;53(10):3954-63. doi: 10.1021/jm901785w. J Med Chem. 2010. PMID: 20408530
New fluoro derivatives of the pyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide system: evaluation of fluorine binding properties in the benzodiazepine site on γ-aminobutyrric acid type A (GABA(A)) receptor. Design, synthesis, biological, and molecular modeling investigation.
Guerrini G, Ciciani G, Bruni F, Selleri S, Guarino C, Melani F, Montali M, Daniele S, Martini C, Ghelardini C, Norcini M, Ciattini S, Costanzo A. Guerrini G, et al. Among authors: martini c. J Med Chem. 2010 Nov 11;53(21):7532-48. doi: 10.1021/jm1001887. J Med Chem. 2010. PMID: 20939501
New 3-, 8-disubstituted pyrazolo[5,1-c][1,2,4]benzotriazines useful for studying the interaction with the HBp-3 area (hydrogen bond point area) in the benzodiazepine site on the γ-aminobutyric acid type A (GABAA) receptor.
Guerrini G, Ciciani G, Bruni F, Selleri S, Melani F, Daniele S, Martini C, Costanzo A. Guerrini G, et al. Among authors: martini c. Bioorg Med Chem. 2011 May 15;19(10):3074-85. doi: 10.1016/j.bmc.2011.04.009. Epub 2011 Apr 12. Bioorg Med Chem. 2011. PMID: 21530274
New insight into the central benzodiazepine receptor-ligand interactions: design, synthesis, biological evaluation, and molecular modeling of 3-substituted 6-phenyl-4H-imidazo[1,5-a][1,4]benzodiazepines and related compounds.
Anzini M, Valenti S, Braile C, Cappelli A, Vomero S, Alcaro S, Ortuso F, Marinelli L, Limongelli V, Novellino E, Betti L, Giannaccini G, Lucacchini A, Daniele S, Martini C, Ghelardini C, Di Cesare Mannelli L, Giorgi G, Mascia MP, Biggio G. Anzini M, et al. Among authors: martini c. J Med Chem. 2011 Aug 25;54(16):5694-711. doi: 10.1021/jm2001597. Epub 2011 Jul 27. J Med Chem. 2011. PMID: 21751815
1,031 results