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Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease.
Eur J Med Chem. 2023 Jan 15;246:114925. doi: 10.1016/j.ejmech.2022.114925. Epub 2022 Nov 15.
Eur J Med Chem. 2023.
PMID: 36459758
Free article.
2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling.
Ferreira RAA, Junior COR, Martinez PDG, Koovits PJ, Soares BM, Ferreira LLG, Michelan-Duarte S, Chelucci RC, Andricopulo AD, Galuppo MK, Uliana SRB, Matheeussen A, Caljon G, Maes L, Campbell S, Kratz JM, Mowbray CE, Dias LC.
Ferreira RAA, et al. Among authors: martinez pdg.
PLoS Negl Trop Dis. 2021 Feb 22;15(2):e0009196. doi: 10.1371/journal.pntd.0009196. eCollection 2021 Feb.
PLoS Negl Trop Dis. 2021.
PMID: 33617566
Free PMC article.
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From rational design to serendipity: Discovery of novel thiosemicarbazones as potent trypanocidal compounds.
Braga SFP, Santos VC, Vieira RP, Silva EBD, Monti L, Krake SH, Martinez PDG, Dias LC, Caffrey CR, Siqueira-Neto JL, de Oliveira RB, Ferreira RS.
Braga SFP, et al. Among authors: martinez pdg.
Eur J Med Chem. 2022 Dec 15;244:114876. doi: 10.1016/j.ejmech.2022.114876. Epub 2022 Oct 27.
Eur J Med Chem. 2022.
PMID: 36343429
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2,3,8-Trisubstituted Quinolines with Antimalarial Activity.
Martinez PDG, Krake SH, Poggi ML, Campbell SF, Willis PA, Dias LC.
Martinez PDG, et al.
An Acad Bras Cienc. 2018 May 21;90(1 Suppl 2):1215-1231. doi: 10.1590/0001-3765201820170820. Print 2018.
An Acad Bras Cienc. 2018.
PMID: 29791525
Free article.
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Novel inhibitors of Plasmodium falciparum based on 2,5-disubstituted furans.
Krake SH, Martinez PDG, McLaren J, Ryan E, Chen G, White K, Charman SA, Campbell S, Willis P, Dias LC.
Krake SH, et al. Among authors: martinez pdg.
Eur J Med Chem. 2017 Jan 27;126:929-936. doi: 10.1016/j.ejmech.2016.12.024. Epub 2016 Dec 11.
Eur J Med Chem. 2017.
PMID: 28002775
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Synthesis of indazoles by the [3+2] cycloaddition of diazo compounds with arynes and subsequent acyl migration.
Liu Z, Shi F, Martinez PD, Raminelli C, Larock RC.
Liu Z, et al.
J Org Chem. 2008 Jan 4;73(1):219-26. doi: 10.1021/jo702062n. Epub 2007 Dec 8.
J Org Chem. 2008.
PMID: 18067316
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