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A very-high-energy component deep in the γ-ray burst afterglow.
Abdalla H, Adam R, Aharonian F, Ait Benkhali F, Angüner EO, Arakawa M, Arcaro C, Armand C, Ashkar H, Backes M, Barbosa Martins V, Barnard M, Becherini Y, Berge D, Bernlöhr K, Bissaldi E, Blackwell R, Böttcher M, Boisson C, Bolmont J, Bonnefoy S, Bregeon J, Breuhaus M, Brun F, Brun P, Bryan M, Büchele M, Bulik T, Bylund T, Capasso M, Caroff S, Carosi A, Casanova S, Cerruti M, Chand T, Chandra S, Chen A, Colafrancesco S, Curyło M, Davids ID, Deil C, Devin J, deWilt P, Dirson L, Djannati-Ataï A, Dmytriiev A, Donath A, Doroshenko V, Dyks J, Egberts K, Emery G, Ernenwein JP, Eschbach S, Feijen K, Fegan S, Fiasson A, Fontaine G, Funk S, Füßling M, Gabici S, Gallant YA, Gaté F, Giavitto G, Giunti L, Glawion D, Glicenstein JF, Gottschall D, Grondin MH, Hahn J, Haupt M, Heinzelmann G, Henri G, Hermann G, Hinton JA, Hofmann W, Hoischen C, Holch TL, Holler M, Horns D, Huber D, Iwasaki H, Jamrozy M, Jankowsky D, Jankowsky F, Jardin-Blicq A, Jung-Richardt I, Kastendieck MA, Katarzyński K, Katsuragawa M, Katz U, Khangulyan D, Khélifi B, King J, Klepser S, Kluźniak W, Komin N, Kosack K, Kostunin D, Kreter M, Lamanna G, Lemière A, Lemoine-Goumard M, Lenain JP, Leser E, Levy C, Lohse T, Lypova I, … See abstract for full author list ➔ Abdalla H, et al. Among authors: mares a. Nature. 2019 Nov;575(7783):464-467. doi: 10.1038/s41586-019-1743-9. Epub 2019 Nov 20. Nature. 2019. PMID: 31748724
Revealing x-ray and gamma ray temporal and spectral similarities in the GRB 190829A afterglow.
H.E.S.S. Collaboration; Abdalla H, Aharonian F, Ait Benkhali F, Angüner EO, Arcaro C, Armand C, Armstrong T, Ashkar H, Backes M, Baghmanyan V, Barbosa Martins V, Barnacka A, Barnard M, Becherini Y, Berge D, Bernlöhr K, Bi B, Bissaldi E, Böttcher M, Boisson C, Bolmont J, de Bony de Lavergne M, Breuhaus M, Brun F, Brun P, Bryan M, Büchele M, Bulik T, Bylund T, Caroff S, Carosi A, Casanova S, Chand T, Chandra S, Chen A, Cotter G, Curyło M, Damascene Mbarubucyeye J, Davids ID, Davies J, Deil C, Devin J, Dirson L, Djannati-Ataï A, Dmytriiev A, Donath A, Doroshenko V, Dreyer L, Duffy C, Dyks J, Egberts K, Eichhorn F, Einecke S, Emery G, Ernenwein JP, Feijen K, Fegan S, Fiasson A, Fichet de Clairfontaine G, Fontaine G, Funk S, Füßling M, Gabici S, Gallant YA, Giavitto G, Giunti L, Glawion D, Glicenstein JF, Grondin MH, Hahn J, Haupt M, Hermann G, Hinton JA, Hofmann W, Hoischen C, Holch TL, Holler M, Hörbe M, Horns D, Huber D, Jamrozy M, Jankowsky D, Jankowsky F, Jardin-Blicq A, Joshi V, Jung-Richardt I, Kasai E, Kastendieck MA, Katarzyński K, Katz U, Khangulyan D, Khélifi B, Klepser S, Kluźniak W, Komin N, Konno R, Kosack K, Kostunin D, Kreter M, Lamanna G, Lemière A, Lemoine-Goumard M, … See abstract for full author list ➔ H.E.S.S. Collaboration, et al. Among authors: mares a. Science. 2021 Jun 4;372(6546):1081-1085. doi: 10.1126/science.abe8560. Science. 2021. PMID: 34083487
Catalytic in vivo protein knockdown by small-molecule PROTACs.
Bondeson DP, Mares A, Smith IE, Ko E, Campos S, Miah AH, Mulholland KE, Routly N, Buckley DL, Gustafson JL, Zinn N, Grandi P, Shimamura S, Bergamini G, Faelth-Savitski M, Bantscheff M, Cox C, Gordon DA, Willard RR, Flanagan JJ, Casillas LN, Votta BJ, den Besten W, Famm K, Kruidenier L, Carter PS, Harling JD, Churcher I, Crews CM. Bondeson DP, et al. Among authors: mares a. Nat Chem Biol. 2015 Aug;11(8):611-7. doi: 10.1038/nchembio.1858. Epub 2015 Jun 10. Nat Chem Biol. 2015. PMID: 26075522 Free PMC article.
Extended pharmacodynamic responses observed upon PROTAC-mediated degradation of RIPK2.
Mares A, Miah AH, Smith IED, Rackham M, Thawani AR, Cryan J, Haile PA, Votta BJ, Beal AM, Capriotti C, Reilly MA, Fisher DT, Zinn N, Bantscheff M, MacDonald TT, Vossenkamper A, Dace P, Churcher I, Benowitz AB, Watt G, Denyer J, Scott-Stevens P, Harling JD. Mares A, et al. Commun Biol. 2020 Mar 20;3(1):140. doi: 10.1038/s42003-020-0868-6. Commun Biol. 2020. PMID: 32198438 Free PMC article.
Optimization of a Series of RIPK2 PROTACs.
Miah AH, Smith IED, Rackham M, Mares A, Thawani AR, Nagilla R, Haile PA, Votta BJ, Gordon LJ, Watt G, Denyer J, Fisher DT, Dace P, Giffen P, Goncalves A, Churcher I, Scott-Stevens P, Harling JD. Miah AH, et al. Among authors: mares a. J Med Chem. 2021 Sep 9;64(17):12978-13003. doi: 10.1021/acs.jmedchem.1c01118. Epub 2021 Aug 25. J Med Chem. 2021. PMID: 34432979
226 results