Malherbe P - Search Results

1

Positive allosteric modulation of GABAB receptors ameliorates sensorimotor gating in rodent models.

Frau R, Bini V, Pillolla G, Malherbe P, Pardu A, Thomas AW, Devoto P, Bortolato M. Frau R, et al. Among authors: malherbe p. CNS Neurosci Ther. 2014 Jul;20(7):679-84. doi: 10.1111/cns.12261. Epub 2014 Apr 7. CNS Neurosci Ther. 2014. PMID: 24703381 Free PMC article.

2

The positive allosteric modulator of the GABA(B) receptor, rac-BHFF, suppresses alcohol self-administration.

Maccioni P, Thomas AW, Carai MA, Gessa GL, Malherbe P, Colombo G. Maccioni P, et al. Among authors: malherbe p. Drug Alcohol Depend. 2010 Jun 1;109(1-3):96-103. doi: 10.1016/j.drugalcdep.2009.12.019. Epub 2010 Jan 20. Drug Alcohol Depend. 2010. PMID: 20089372

3

Reduction of alcohol intake by the positive allosteric modulator of the GABA(B) receptor, rac-BHFF, in alcohol-preferring rats.

Loi B, Maccioni P, Lobina C, Carai MA, Gessa GL, Thomas AW, Malherbe P, Colombo G. Loi B, et al. Among authors: malherbe p. Alcohol. 2013 Feb;47(1):69-73. doi: 10.1016/j.alcohol.2012.11.002. Epub 2012 Dec 6. Alcohol. 2013. PMID: 23218664

4

Inhibition of alcohol self-administration by positive allosteric modulators of the GABAB receptor in rats: lack of tolerance and potentiation of baclofen.

Maccioni P, Vargiolu D, Thomas AW, Malherbe P, Mugnaini C, Corelli F, Leite-Morris KA, Gessa GL, Colombo G. Maccioni P, et al. Among authors: malherbe p. Psychopharmacology (Berl). 2015 May;232(10):1831-41. doi: 10.1007/s00213-014-3815-8. Epub 2014 Nov 26. Psychopharmacology (Berl). 2015. PMID: 25420609

5

Characterization of (R,S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one as a positive allosteric modulator of GABAB receptors.

Malherbe P, Masciadri R, Norcross RD, Knoflach F, Kratzeisen C, Zenner MT, Kolb Y, Marcuz A, Huwyler J, Nakagawa T, Porter RH, Thomas AW, Wettstein JG, Sleight AJ, Spooren W, Prinssen EP. Malherbe P, et al. Br J Pharmacol. 2008 Jun;154(4):797-811. doi: 10.1038/bjp.2008.135. Epub 2008 Apr 21. Br J Pharmacol. 2008. PMID: 18536733 Free PMC article.

6

The positive allosteric GABAB receptor modulator rac-BHFF enhances baclofen-mediated analgesia in neuropathic mice.

Zemoura K, Ralvenius WT, Malherbe P, Benke D. Zemoura K, et al. Among authors: malherbe p. Neuropharmacology. 2016 Sep;108:172-8. doi: 10.1016/j.neuropharm.2016.04.028. Epub 2016 Apr 22. Neuropharmacology. 2016. PMID: 27108932

7

Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX(2) receptor.

Malherbe P, Borroni E, Gobbi L, Knust H, Nettekoven M, Pinard E, Roche O, Rogers-Evans M, Wettstein JG, Moreau JL. Malherbe P, et al. Br J Pharmacol. 2009 Apr;156(8):1326-41. doi: 10.1111/j.1476-5381.2009.00127.x. Br J Pharmacol. 2009. PMID: 19751316 Free PMC article.

8

Characterization of RO4583298 as a novel potent, dual antagonist with in vivo activity at tachykinin NK₁ and NK₃ receptors.

Malherbe P, Knoflach F, Hernandez MC, Hoffmann T, Schnider P, Porter RH, Wettstein JG, Ballard TM, Spooren W, Steward L. Malherbe P, et al. Br J Pharmacol. 2011 Feb;162(4):929-46. doi: 10.1111/j.1476-5381.2010.01096.x. Br J Pharmacol. 2011. PMID: 21039418 Free PMC article.

9

Fenobam: a clinically validated nonbenzodiazepine anxiolytic is a potent, selective, and noncompetitive mGlu5 receptor antagonist with inverse agonist activity.

Porter RH, Jaeschke G, Spooren W, Ballard TM, Büttelmann B, Kolczewski S, Peters JU, Prinssen E, Wichmann J, Vieira E, Mühlemann A, Gatti S, Mutel V, Malherbe P. Porter RH, et al. Among authors: malherbe p. J Pharmacol Exp Ther. 2005 Nov;315(2):711-21. doi: 10.1124/jpet.105.089839. Epub 2005 Jul 22. J Pharmacol Exp Ther. 2005. PMID: 16040814

10

Determination of key amino acids implicated in the actions of allosteric modulation by 3,3'-difluorobenzaldazine on rat mGlu5 receptors.

Mühlemann A, Ward NA, Kratochwil N, Diener C, Fischer C, Stucki A, Jaeschke G, Malherbe P, Porter RH. Mühlemann A, et al. Among authors: malherbe p. Eur J Pharmacol. 2006 Jan 4;529(1-3):95-104. doi: 10.1016/j.ejphar.2005.11.008. Epub 2005 Dec 13. Eur J Pharmacol. 2006. PMID: 16352303

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