Makara GM - Search Results

1

Label-free high-throughput screening via mass spectrometry: a single cystathionine quantitative method for multiple applications.

Holt TG, Choi BK, Geoghagen NS, Jensen KK, Luo Q, LaMarr WA, Makara GM, Malkowitz L, Ozbal CC, Xiong Y, Dufresne C, Luo MJ. Holt TG, et al. Among authors: makara gm. Assay Drug Dev Technol. 2009 Oct;7(5):495-506. doi: 10.1089/adt.2009.0200. Assay Drug Dev Technol. 2009. PMID: 19715455

2

Improving success rates for lead generation using affinity binding technologies.

Makara GM, Athanasopoulos J. Makara GM, et al. Curr Opin Biotechnol. 2005 Dec;16(6):666-73. doi: 10.1016/j.copbio.2005.10.007. Epub 2005 Oct 28. Curr Opin Biotechnol. 2005. PMID: 16257522 Free PMC article. Review.

3

On sampling of fragment space.

Makara GM. Makara GM. J Med Chem. 2007 Jul 12;50(14):3214-21. doi: 10.1021/jm0700316. Epub 2007 Jun 14. J Med Chem. 2007. PMID: 17567120

4

Hit discovery and hit-to-lead approaches.

Keseru GM, Makara GM. Keseru GM, et al. Among authors: makara gm. Drug Discov Today. 2006 Aug;11(15-16):741-8. doi: 10.1016/j.drudis.2006.06.016. Drug Discov Today. 2006. PMID: 16846802 Review.

5

New developments in chemical library synthesis. Norbornenyl tags for use in phase-switching, sequestration, capture-release and soluble support applications.

Flynn DL, Hanson PR, Berk SC, Makara GM. Flynn DL, et al. Among authors: makara gm. Curr Opin Drug Discov Devel. 2002 Jul;5(4):571-9. Curr Opin Drug Discov Devel. 2002. PMID: 12197315 Review.

6

Recent advances in chemical library synthesis methodology.

Flynn DL, Berk SC, Makara GM. Flynn DL, et al. Among authors: makara gm. Curr Opin Drug Discov Devel. 2002 Jul;5(4):580-93. Curr Opin Drug Discov Devel. 2002. PMID: 12197316 Review.

7

Synthesis and modeling studies with monocyclic analogues of mycophenolic acid.

Anderson WK, Boehm TL, Makara GM, Swann RT. Anderson WK, et al. Among authors: makara gm. J Med Chem. 1996 Jan 5;39(1):46-55. doi: 10.1021/jm9501339. J Med Chem. 1996. PMID: 8568826

8

Nuclear magnetic resonance and molecular modeling study on mycophenolic acid: implications for binding to inosine monophosphate dehydrogenase.

Makara GM, Keserû GM, Kajtár-Peredy M, Anderson WK. Makara GM, et al. J Med Chem. 1996 Mar 15;39(6):1236-42. doi: 10.1021/jm950600m. J Med Chem. 1996. PMID: 8632430

9

Identification of a small molecule nonpeptide active site beta-secretase inhibitor that displays a nontraditional binding mode for aspartyl proteases.

Coburn CA, Stachel SJ, Li YM, Rush DM, Steele TG, Chen-Dodson E, Holloway MK, Xu M, Huang Q, Lai MT, DiMuzio J, Crouthamel MC, Shi XP, Sardana V, Chen Z, Munshi S, Kuo L, Makara GM, Annis DA, Tadikonda PK, Nash HM, Vacca JP, Wang T. Coburn CA, et al. Among authors: makara gm. J Med Chem. 2004 Dec 2;47(25):6117-9. doi: 10.1021/jm049388p. J Med Chem. 2004. PMID: 15566281

10

Measuring molecular similarity and diversity: total pharmacophore diversity.

Makara GM. Makara GM. J Med Chem. 2001 Oct 25;44(22):3563-71. doi: 10.1021/jm010036h. J Med Chem. 2001. PMID: 11606120

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