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Pt(IV) Prodrugs with Non-Steroidal Anti-inflammatory Drugs in the Axial Position.
Spector DV, Pavlov KG, Akasov RA, Vaneev AN, Erofeev AS, Gorelkin PV, Nikitina VN, Lopatukhina EV, Semkina AS, Vlasova KY, Skvortsov DA, Roznyatovsky VA, Ul'yanovskiy NV, Pikovskoi II, Sypalov SA, Garanina AS, Vodopyanov SS, Abakumov MA, Volodina YL, Markova AA, Petrova AS, Mazur DM, Sakharov DA, Zyk NV, Beloglazkina EK, Majouga AG, Krasnovskaya OO. Spector DV, et al. Among authors: majouga ag. J Med Chem. 2022 Jun 23;65(12):8227-8244. doi: 10.1021/acs.jmedchem.1c02136. Epub 2022 Jun 8. J Med Chem. 2022. PMID: 35675651
Mixed valence copper(I,II) binuclear complexes with unexpected structure: synthesis, biological properties and anticancer activity.
Majouga AG, Zvereva MI, Rubtsova MP, Skvortsov DA, Mironov AV, Azhibek DM, Krasnovskaya OO, Gerasimov VM, Udina AV, Vorozhtsov NI, Beloglazkina EK, Agron L, Mikhina LV, Tretyakova AV, Zyk NV, Zefirov NS, Kabanov AV, Dontsova OA. Majouga AG, et al. J Med Chem. 2014 Jul 24;57(14):6252-8. doi: 10.1021/jm500154f. Epub 2014 Jul 8. J Med Chem. 2014. PMID: 24950478
Enzyme-functionalized gold-coated magnetite nanoparticles as novel hybrid nanomaterials: synthesis, purification and control of enzyme function by low-frequency magnetic field.
Majouga A, Sokolsky-Papkov M, Kuznetsov A, Lebedev D, Efremova M, Beloglazkina E, Rudakovskaya P, Veselov M, Zyk N, Golovin Y, Klyachko N, Kabanov A. Majouga A, et al. Colloids Surf B Biointerfaces. 2015 Jan 1;125:104-9. doi: 10.1016/j.colsurfb.2014.11.012. Epub 2014 Nov 20. Colloids Surf B Biointerfaces. 2015. PMID: 25460600
Design, synthesis and biological evaluation of novel potent MDM2/p53 small-molecule inhibitors.
Ivanenkov YA, Vasilevski SV, Beloglazkina EK, Kukushkin ME, Machulkin AE, Veselov MS, Chufarova NV, Chernyaginab ES, Vanzcool AS, Zyk NV, Skvortsov DA, Khutornenko AA, Rusanov AL, Tonevitsky AG, Dontsova OA, Majouga AG. Ivanenkov YA, et al. Among authors: majouga ag. Bioorg Med Chem Lett. 2015 Jan 15;25(2):404-9. doi: 10.1016/j.bmcl.2014.09.070. Epub 2014 Oct 2. Bioorg Med Chem Lett. 2015. PMID: 25479770
Development of bacteriochlorophyll a-based near-infrared photosensitizers conjugated to gold nanoparticles for photodynamic therapy of cancer.
Pantiushenko IV, Rudakovskaya PG, Starovoytova AV, Mikhaylovskaya AA, Abakumov MA, Kaplan MA, Tsygankov AA, Majouga AG, Grin MA, Mironov AF. Pantiushenko IV, et al. Among authors: majouga ag. Biochemistry (Mosc). 2015 Jun;80(6):752-62. doi: 10.1134/S0006297915060103. Biochemistry (Mosc). 2015. PMID: 26531020 Free article. Review.
Synthesis, isomerization and biological activity of novel 2-selenohydantoin derivatives.
Ivanenkov YA, Veselov MS, Rezekin IG, Skvortsov DA, Sandulenko YB, Polyakova MV, Bezrukov DS, Vasilevsky SV, Kukushkin ME, Moiseeva AA, Finko AV, Koteliansky VE, Klyachko NL, Filatova LA, Beloglazkina EK, Zyk NV, Majouga AG. Ivanenkov YA, et al. Among authors: majouga ag. Bioorg Med Chem. 2016 Feb 15;24(4):802-11. doi: 10.1016/j.bmc.2015.12.050. Epub 2016 Jan 2. Bioorg Med Chem. 2016. PMID: 26780833
Small-molecule PSMA ligands. Current state, SAR and perspectives.
Machulkin AE, Ivanenkov YA, Aladinskaya AV, Veselov MS, Aladinskiy VA, Beloglazkina EK, Koteliansky VE, Shakhbazyan AG, Sandulenko YB, Majouga AG. Machulkin AE, et al. Among authors: majouga ag. J Drug Target. 2016 Sep;24(8):679-93. doi: 10.3109/1061186X.2016.1154564. Epub 2016 Mar 10. J Drug Target. 2016. PMID: 26887438 Review.
Identification of Novel Small-Molecule ASGP-R Ligands.
Majouga AG, Ivanenkov YA, Veselov MS, Lopuhov AV, Maklakova SV, Beloglazkina EK, Binevski PV, Klyachko NL, Sandulenko YB, Galkina NY, Koteliansky VE. Majouga AG, et al. Curr Drug Deliv. 2016;13(8):1303-1312. doi: 10.2174/1567201813666160719144651. Curr Drug Deliv. 2016. PMID: 27440073
122 results