Mader P - Search Results

1

Crystal structure of native α-L-rhamnosidase from Aspergillus terreus.

Pachl P, Škerlová J, Šimčíková D, Kotik M, Křenková A, Mader P, Brynda J, Kapešová J, Křen V, Otwinowski Z, Řezáčová P. Pachl P, et al. Among authors: mader p. Acta Crystallogr D Struct Biol. 2018 Nov 1;74(Pt 11):1078-1084. doi: 10.1107/S2059798318013049. Epub 2018 Oct 29. Acta Crystallogr D Struct Biol. 2018. PMID: 30387766

2

Structural basis for the interaction between carbonic anhydrase and 1,2,3,4-tetrahydroisoquinolin-2-ylsulfonamides.

Mader P, Brynda J, Gitto R, Agnello S, Pachl P, Supuran CT, Chimirri A, Řezáčová P. Mader P, et al. J Med Chem. 2011 Apr 14;54(7):2522-6. doi: 10.1021/jm2000213. Epub 2011 Mar 11. J Med Chem. 2011. PMID: 21395315

3

Carborane-based carbonic anhydrase inhibitors: insight into CAII/CAIX specificity from a high-resolution crystal structure, modeling, and quantum chemical calculations.

Mader P, Pecina A, Cígler P, Lepšík M, Šícha V, Hobza P, Grüner B, Fanfrlík J, Brynda J, Řezáčová P. Mader P, et al. Biomed Res Int. 2014;2014:389869. doi: 10.1155/2014/389869. Epub 2014 Sep 18. Biomed Res Int. 2014. PMID: 25309911 Free PMC article.

4

QM/MM calculations reveal the different nature of the interaction of two carborane-based sulfamide inhibitors of human carbonic anhydrase II.

Pecina A, Lepšík M, Řezáč J, Brynda J, Mader P, Řezáčová P, Hobza P, Fanfrlík J. Pecina A, et al. Among authors: mader p. J Phys Chem B. 2013 Dec 19;117(50):16096-104. doi: 10.1021/jp410216m. Epub 2013 Dec 11. J Phys Chem B. 2013. PMID: 24289143

5

Stabilization of antibody structure upon association to a human carbonic anhydrase IX epitope studied by X-ray crystallography, microcalorimetry, and molecular dynamics simulations.

Král V, Mader P, Collard R, Fábry M, Horejsí M, Rezácová P, Kozísek M, Závada J, Sedlácek J, Rulísek L, Brynda J. Král V, et al. Among authors: mader p. Proteins. 2008 May 15;71(3):1275-87. doi: 10.1002/prot.21821. Proteins. 2008. PMID: 18041760

6

Carborane-based carbonic anhydrase inhibitors.

Brynda J, Mader P, Šícha V, Fábry M, Poncová K, Bakardiev M, Grüner B, Cígler P, Řezáčová P. Brynda J, et al. Among authors: mader p. Angew Chem Int Ed Engl. 2013 Dec 16;52(51):13760-3. doi: 10.1002/anie.201307583. Epub 2013 Nov 4. Angew Chem Int Ed Engl. 2013. PMID: 24307504

7

Synthesis, structure-activity relationship studies, and X-ray crystallographic analysis of arylsulfonamides as potent carbonic anhydrase inhibitors.

Gitto R, Damiano FM, Mader P, De Luca L, Ferro S, Supuran CT, Vullo D, Brynda J, Rezáčová P, Chimirri A. Gitto R, et al. Among authors: mader p. J Med Chem. 2012 Apr 26;55(8):3891-9. doi: 10.1021/jm300112w. Epub 2012 Apr 6. J Med Chem. 2012. PMID: 22443141

8

Identification of 3,4-Dihydroisoquinoline-2(1H)-sulfonamides as potent carbonic anhydrase inhibitors: synthesis, biological evaluation, and enzyme--ligand X-ray studies.

Gitto R, Agnello S, Ferro S, De Luca L, Vullo D, Brynda J, Mader P, Supuran CT, Chimirri A. Gitto R, et al. Among authors: mader p. J Med Chem. 2010 Mar 25;53(6):2401-8. doi: 10.1021/jm9014026. J Med Chem. 2010. PMID: 20170095

9

Identification of carbonic anhydrase I immunodominant epitopes recognized by specific autoantibodies which indicate an improved prognosis in patients with malignancy after autologous stem cell transplantation.

Skultety L, Jankovicova B, Svobodova Z, Mader P, Rezacova P, Dubrovcakova M, Lakota J, Bilkova Z. Skultety L, et al. Among authors: mader p. J Proteome Res. 2010 Oct 1;9(10):5171-9. doi: 10.1021/pr1004778. J Proteome Res. 2010. PMID: 20681519

10

Discovery and Structural Characterization of Small Molecule Binders of the Human CTLH E3 Ligase Subunit GID4.

Chana CK, Maisonneuve P, Posternak G, Grinberg NGA, Poirson J, Ona SM, Ceccarelli DF, Mader P, St-Cyr DJ, Pau V, Kurinov I, Tang X, Deng D, Cui W, Su W, Kuai L, Soll R, Tyers M, Röst HL, Batey RA, Taipale M, Gingras AC, Sicheri F. Chana CK, et al. Among authors: mader p. J Med Chem. 2022 Oct 13;65(19):12725-12746. doi: 10.1021/acs.jmedchem.2c00509. Epub 2022 Sep 18. J Med Chem. 2022. PMID: 36117290 Free PMC article.

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