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Differential expression in humans of the viral entry receptor ACE2 compared with the short deltaACE2 isoform lacking SARS-CoV-2 binding sites.
Sci Rep. 2021 Dec 21;11(1):24336. doi: 10.1038/s41598-021-03731-9.
Sci Rep. 2021.
PMID: 34934117
Free PMC article.
International Union of Basic and Clinical Pharmacology. CVII. Structure and Pharmacology of the Apelin Receptor with a Recommendation that Elabela/Toddler Is a Second Endogenous Peptide Ligand.
Read C, Nyimanu D, Williams TL, Huggins DJ, Sulentic P, Macrae RGC, Yang P, Glen RC, Maguire JJ, Davenport AP.
Read C, et al. Among authors: macrae rgc.
Pharmacol Rev. 2019 Oct;71(4):467-502. doi: 10.1124/pr.119.017533.
Pharmacol Rev. 2019.
PMID: 31492821
Free PMC article.
Review.
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THE CONCISE GUIDE TO PHARMACOLOGY 2019/20: G protein-coupled receptors.
Alexander SPH, Christopoulos A, Davenport AP, Kelly E, Mathie A, Peters JA, Veale EL, Armstrong JF, Faccenda E, Harding SD, Pawson AJ, Sharman JL, Southan C, Davies JA; CGTP Collaborators.
Alexander SPH, et al.
Br J Pharmacol. 2019 Dec;176 Suppl 1(Suppl 1):S21-S141. doi: 10.1111/bph.14748.
Br J Pharmacol. 2019.
PMID: 31710717
Free PMC article.
Review.
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Human embryonic stem cell-derived cardiomyocyte platform screens inhibitors of SARS-CoV-2 infection.
Williams TL, Colzani MT, Macrae RGC, Robinson EL, Bloor S, Greenwood EJD, Zhan JR, Strachan G, Kuc RE, Nyimanu D, Maguire JJ, Lehner PJ, Sinha S, Davenport AP.
Williams TL, et al. Among authors: macrae rgc.
Commun Biol. 2021 Jul 29;4(1):926. doi: 10.1038/s42003-021-02453-y.
Commun Biol. 2021.
PMID: 34326460
Free PMC article.
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THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors.
Alexander SP, Christopoulos A, Davenport AP, Kelly E, Mathie A, Peters JA, Veale EL, Armstrong JF, Faccenda E, Harding SD, Pawson AJ, Southan C, Davies JA, Abbracchio MP, Alexander W, Al-Hosaini K, Bäck M, Barnes NM, Bathgate R, Beaulieu JM, Bernstein KE, Bettler B, Birdsall NJM, Blaho V, Boulay F, Bousquet C, Bräuner-Osborne H, Burnstock G, Caló G, Castaño JP, Catt KJ, Ceruti S, Chazot P, Chiang N, Chini B, Chun J, Cianciulli A, Civelli O, Clapp LH, Couture R, Csaba Z, Dahlgren C, Dent G, Singh KD, Douglas SD, Dournaud P, Eguchi S, Escher E, Filardo EJ, Fong T, Fumagalli M, Gainetdinov RR, Gasparo M, Gerard C, Gershengorn M, Gobeil F, Goodfriend TL, Goudet C, Gregory KJ, Gundlach AL, Hamann J, Hanson J, Hauger RL, Hay DL, Heinemann A, Hollenberg MD, Holliday ND, Horiuchi M, Hoyer D, Hunyady L, Husain A, IJzerman AP, Inagami T, Jacobson KA, Jensen RT, Jockers R, Jonnalagadda D, Karnik S, Kaupmann K, Kemp J, Kennedy C, Kihara Y, Kitazawa T, Kozielewicz P, Kreienkamp HJ, Kukkonen JP, Langenhan T, Leach K, Lecca D, Lee JD, Leeman SE, Leprince J, Li XX, Williams TL, Lolait SJ, Lupp A, Macrae R, Maguire J, Mazella J, McArdle CA, Melmed S, Michel MC, Miller LJ, Mitolo V, Mouillac B, Mül…
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Alexander SP, et al.
Br J Pharmacol. 2021 Oct;178 Suppl 1:S27-S156. doi: 10.1111/bph.15538.
Br J Pharmacol. 2021.
PMID: 34529832
Free article.
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Inducible apelin receptor knockdown reduces differentiation efficiency and contractility of hESC-derived cardiomyocytes.
Macrae RGC, Colzani MT, Williams TL, Bayraktar S, Kuc RE, Pullinger AL, Bernard WG, Robinson EL, Davenport EE, Maguire JJ, Sinha S, Davenport AP.
Macrae RGC, et al.
Cardiovasc Res. 2023 Mar 31;119(2):587-598. doi: 10.1093/cvr/cvac065.
Cardiovasc Res. 2023.
PMID: 36239923
Free PMC article.
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A phenotypic screen of Marfan syndrome iPSC-derived vascular smooth muscle cells uncovers GSK3β as a new target.
Davaapil H, McNamara M, Granata A, Macrae RGC, Hirano M, Fitzek M, Aragon-Martin JA, Child A, Smith DM, Sinha S.
Davaapil H, et al. Among authors: macrae rgc.
Stem Cell Reports. 2023 Feb 14;18(2):555-569. doi: 10.1016/j.stemcr.2022.12.014. Epub 2023 Jan 19.
Stem Cell Reports. 2023.
PMID: 36669494
Free PMC article.
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Expanding the apelin receptor pharmacological toolbox using novel fluorescent ligands.
Williams TL, Macrae RGC, Kuc RE, Brown AJH, Maguire JJ, Davenport AP.
Williams TL, et al. Among authors: macrae rgc.
Front Endocrinol (Lausanne). 2023 Mar 9;14:1139121. doi: 10.3389/fendo.2023.1139121. eCollection 2023.
Front Endocrinol (Lausanne). 2023.
PMID: 36967803
Free PMC article.
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